# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4580164 | 2 | Ratio | > | 4 | ALA4385847 | ||||||
2. | ALA4580164 | 2 | Cmax | = | 294 | ng/ml | ALA4385815 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
3. | ALA4580164 | 2 | IC50 | > | 10000 | nM | ALA4385804 | nM | Homo sapiens | |||
4. | ALA4580164 | 2 | IC50 | = | 4010 | nM | ALA4385809 | 5.40 | nM | Homo sapiens | ||
5. | ALA4580164 | 2 | IC50 | = | 4830 | nM | ALA4385811 | 5.32 | nM | Homo sapiens | ||
6. | ALA4580164 | 2 | IC50 | > | 10000 | nM | ALA4385812 | nM | Homo sapiens | |||
7. | ALA4580164 | 2 | IC50 | = | 8.7 | nM | ALA4385807 | 8.06 | nM | Homo sapiens | ||
8. | ALA4580164 | 2 | Activity | 0 | ALA4385845 | Active | Mus musculus | |||||
9. | ALA4580164 | 2 | Activity | 0 | ALA4385844 | Active | Mus musculus | |||||
10. | ALA4580164 | 2 | Activity | 0 | ALA4385843 | Active | Mus musculus | |||||
11. | ALA4580164 | 2 | Activity | 0 | ALA4385842 | Active | Mus musculus | |||||
12. | ALA4580164 | 2 | Time | = | 22.04 | s | ALA4385841 | hr | Mus musculus | |||
13. | ALA4580164 | 2 | Time | = | 34.55 | s | ALA4385840 | hr | Mus musculus | |||
14. | ALA4580164 | 2 | Activity | > | 1.5 | g/Kg | ALA4385787 | g/Kg | ||||
15. | ALA4580164 | 2 | IC50 | > | 10 | uM | ALA4385786 | nM | Homo sapiens | |||
16. | ALA4580164 | 2 | IC50 | > | 10 | uM | ALA4385839 | nM | Homo sapiens | |||
17. | ALA4580164 | 2 | IC50 | > | 10 | uM | ALA4385838 | nM | Homo sapiens | |||
18. | ALA4580164 | 2 | IC50 | > | 10 | uM | ALA4385837 | nM | Homo sapiens | |||
19. | ALA4580164 | 2 | IC50 | > | 10 | uM | ALA4385836 | nM | Homo sapiens | |||
20. | ALA4580164 | 2 | PPB | = | 78 | % | ALA4385833 | % |