| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4580469 | 26b | Kinetic_solubility | < | 5 | uM | ALA4384260 | nM | ||||
| 2. | ALA4580469 | 26b | log(Kinetic_solubility) | < | -5 | ALA4384260 | ||||||
| 3. | ALA4580469 | 26b | Kinetic_solubility | < | 5 | uM | ALA4384259 | nM | ||||
| 4. | ALA4580469 | 26b | log(Kinetic_solubility) | < | -5 | ALA4384259 | ||||||
| 5. | ALA4580469 | 26b | Ratio | = | 0.95 | ALA4384258 | ||||||
| 6. | ALA4580469 | 26b | Drug recovery | = | 97 | % | ALA4384257 | % | ||||
| 7. | ALA4580469 | 26b | Drug recovery | = | 83 | % | ALA4384256 | % | ||||
| 8. | ALA4580469 | 26b | Papp | = | 20 | 10'-6 cm/s | ALA4384255 | 10'-6 cm/s | ||||
| 9. | ALA4580469 | 26b | Papp | = | 21 | 10'-6 cm/s | ALA4384254 | 10'-6 cm/s | ||||
| 10. | ALA4580469 | 26b | PPB | = | 99 | % | ALA4384253 | % | ||||
| 11. | ALA4580469 | 26b | Stability | > | 99 | % | ALA4384252 | % | ||||
| 12. | ALA4580469 | 26b | Stability | = | 97 | % | ALA4384251 | % | ||||
| 13. | ALA4580469 | 26b | Stability | = | 3.6 | % | ALA4384250 | % | ||||
| 14. | ALA4580469 | 26b | Stability | = | 92 | % | ALA4384249 | % | ||||
| 15. | ALA4580469 | 26b | IC50 | = | 0.24 | uM | ALA4384236 | 6.62 | nM | Trypanosoma brucei brucei | ||
| 16. | ALA4580469 | 26b | pIC50 | = | 5.7 | ALA4384236 | 5.70 | nM | Trypanosoma brucei brucei | |||
| 17. | ALA4580469 | 26b | MIC | = | 4 | ug ml-1 | ALA4384233 | ug.mL-1 | Mycobacterium tuberculosis | |||
| 18. | ALA4580469 | 26b | MIC=<90 | = | 1 | ug ml-1 | ALA4384231 | ug ml-1 | Mycobacterium tuberculosis | |||
| 19. | ALA4580469 | 26b | pIC50 | = | 5 | ALA4384229 | 5.00 | nM | Entamoeba histolytica | |||
| 20. | ALA4580469 | 26b | IC50 | = | 10 | uM | ALA4384229 | 5.00 | nM | Entamoeba histolytica |
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