# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4580825 | 22 | IC50 | = | 4.9 | uM | ALA4384350 | 5.31 | nM | |||
2. | ALA4580825 | 22 | IC50 | = | 2.9 | uM | ALA4384349 | 5.54 | nM | |||
3. | ALA4580825 | 22 | Activity | = | 51 | % | ALA4384347 | % | ||||
4. | ALA4580825 | 22 | Activity | = | 140 | % | ALA4384345 | % | ||||
5. | ALA4580825 | 22 | INH | 0 | ALA4384343 | Not Active | % | |||||
6. | ALA4580825 | 22 | INH | 0 | ALA4384341 | Not Active | % | |||||
7. | ALA4580825 | 22 | Kinetic_solubility | = | 4.2 | 10'-6mg/ml | ALA4384339 | ug.mL-1 | ||||
8. | ALA4580825 | 22 | Kinetic_solubility | = | 2.4 | 10'-3mg/ml | ALA4384338 | ug.mL-1 | ||||
9. | ALA4580825 | 22 | CLH | = | 22 | ml/min | ALA4384337 | ml/min | ||||
10. | ALA4580825 | 22 | t1/2 | = | 31 | min | ALA4384336 | hr | ||||
11. | ALA4580825 | 22 | GI50 | = | 2.2 | uM | ALA4384335 | nM | ||||
12. | ALA4580825 | 22 | EC50 | = | 0.6 | uM | ALA4384334 | 6.22 | nM | Mus musculus | ||
13. | ALA4580825 | 22 | Activity | > | 30000 | % | ALA4384331 | % | Mus musculus | |||
14. | ALA4580825 | 22 | IC50 | = | 0.2 | uM | ALA4384330 | 6.70 | nM | |||
15. | ALA4580825 | 22 | Activity | = | 15000 | % | ALA4384328 | % | Mus musculus | |||
16. | ALA4580825 | 22 | IC50 | = | 0.89 | uM | ALA4384327 | 6.05 | nM | |||
17. | ALA4580825 | 22 | INH | = | 11 | % | ALA4384324 | % |