# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4581366 | 2 | IC50 | = | 38 | nM | ALA4416027 | 7.42 | nM | Homo sapiens | ||
2. | ALA4581366 | 2 | IC50 | = | 12 | nM | ALA4416028 | 7.92 | nM | Homo sapiens | ||
3. | ALA4581366 | 2 | deltaTm | = | 37.5 | degrees C | ALA4416029 | degrees C | Homo sapiens | |||
4. | ALA4581366 | 2 | deltaTm | = | 38 | degrees C | ALA4416030 | degrees C | Homo sapiens | |||
5. | ALA4581366 | 2 | IC50 | = | 25 | nM | ALA4416031 | 7.60 | nM | Homo sapiens | ||
6. | ALA4581366 | 2 | IC50 | = | 14 | nM | ALA4416032 | 7.85 | nM | Homo sapiens | ||
7. | ALA4581366 | 2 | IC50 | = | 28 | nM | ALA4416026 | 7.55 | nM | Homo sapiens | ||
8. | ALA4581366 | 2 | IC50 | = | 9 | nM | ALA4416033 | 8.05 | nM | Homo sapiens | ||
9. | ALA4581366 | 2 | Stability | 0 | ALA4416034 | Stable | % | |||||
10. | ALA4581366 | 2 | solubility | <= | 2 | mM | ALA4416035 | nM | ||||
11. | ALA4581366 | 2 | t1/2 | > | 2 | hr | ALA4416036 | hr | ||||
12. | ALA4581366 | 2 | Activity | 0 | ALA4416037 | Active | Homo sapiens | |||||
13. | ALA4581366 | 2 | Activity | 0 | ALA4416038 | Active | Homo sapiens | |||||
14. | ALA4581366 | 2 | Activity | 0 | ALA4416039 | Active | Homo sapiens | |||||
15. | ALA4581366 | 2 | Activity | 0 | ALA4416040 | Active | Homo sapiens | |||||
16. | ALA4581366 | 2 | Activity | 0 | ALA4416041 | Active | Homo sapiens | |||||
17. | ALA4581366 | 2 | Activity | 0 | ALA4416042 | Not Active | Homo sapiens | |||||
18. | ALA4581366 | 2 | Activity | 0 | ALA4416043 | Not Active | Homo sapiens | |||||
19. | ALA4581366 | 2 | Activity | 0 | ALA4416044 | Dose-dependent effect | Homo sapiens | |||||
20. | ALA4581366 | 2 | Activity | 0 | ALA4416045 | Dose-dependent effect | Homo sapiens |