# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4582879 | 38; UR-AP158 | Ratio Ki | = | 4900 | ALA4397801 | Homo sapiens | |||||
2. | ALA4582879 | 38; UR-AP158 | Ratio Ki | = | 40 | ALA4397800 | Homo sapiens | |||||
3. | ALA4582879 | 38; UR-AP158 | Ratio Ki | = | 1800 | ALA4397799 | Homo sapiens | |||||
4. | ALA4582879 | 38; UR-AP158 | Ratio Ki | = | 45 | ALA4397798 | Homo sapiens | |||||
5. | ALA4582879 | 38; UR-AP158 | pKi | = | 6.53 | ALA4397797 | 6.53 | nM | Homo sapiens | |||
6. | ALA4582879 | 38; UR-AP158 | pKi | = | 8.68 | ALA4397796 | 8.68 | nM | Homo sapiens | |||
7. | ALA4582879 | 38; UR-AP158 | pKi | = | 6.96 | ALA4397795 | 6.96 | nM | Homo sapiens | |||
8. | ALA4582879 | 38; UR-AP158 | pKi | = | 10.2 | ALA4397794 | 10.20 | nM | Homo sapiens | |||
9. | ALA4582879 | 38; UR-AP158 | pKi | = | 8.64 | ALA4397793 | 8.64 | nM | Homo sapiens | |||
10. | ALA4582879 | 38; UR-AP158 | pIC50 | = | 8.75 | ALA4397809 | 8.75 | nM | Homo sapiens | |||
11. | ALA4582879 | 38; UR-AP158 | pIC50 | = | 9.72 | ALA4397808 | 9.72 | nM | Homo sapiens | |||
12. | ALA4582879 | 38; UR-AP158 | pIC50 | = | 7.98 | ALA4397803 | 7.98 | nM | Homo sapiens | |||
13. | ALA4582879 | 38; UR-AP158 | Activity | > | 95 | % | ALA4397810 | % | Homo sapiens | |||
14. | ALA4582879 | 38; UR-AP158 | pKi | = | 10.1 | ALA4397809 | 10.10 | nM | Homo sapiens | |||
15. | ALA4582879 | 38; UR-AP158 | pKi | = | 10.2 | ALA4397808 | 10.20 | nM | Homo sapiens | |||
16. | ALA4582879 | 38; UR-AP158 | Stability | > | 99 | % | ALA4397807 | % | ||||
17. | ALA4582879 | 38; UR-AP158 | Stability | > | 99 | % | ALA4397806 | % | ||||
18. | ALA4582879 | 38; UR-AP158 | Stability | > | 99 | % | ALA4397805 | % | ||||
19. | ALA4582879 | 38; UR-AP158 | Stability | > | 99 | % | ALA4397804 | % | ||||
20. | ALA4582879 | 38; UR-AP158 | INH | 0 | ALA4397803 | Dose-dependent effect | % | Homo sapiens |