# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4583457 | 3g | AUC | = | 140 | uM.hr | ALA4327024 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
2. | ALA4583457 | 3g | F | = | 55 | % | ALA4327028 | % | ||||
3. | ALA4583457 | 3g | F | = | 55 | % | ALA4327027 | % | ||||
4. | ALA4583457 | 3g | t1/2 | = | 6.7 | hr | ALA4327026 | hr | ||||
5. | ALA4583457 | 3g | AUC | = | 79 | uM.hr | ALA4327025 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
6. | ALA4583457 | 3g | Fu | = | 1.5 | % | ALA4327023 | |||||
7. | ALA4583457 | 3g | permeability | = | 712 | nm/s | ALA4327022 | nm/s | ||||
8. | ALA4583457 | 3g | permeability | = | 960 | nm/s | ALA4327021 | nm/s | ||||
9. | ALA4583457 | 3g | Stability | = | 79 | % | ALA4327020 | % | ||||
10. | ALA4583457 | 3g | IC50 | = | 81 | uM | ALA4327019 | 4.09 | nM | Homo sapiens | ||
11. | ALA4583457 | 3g | IC50 | = | 49 | nM | ALA4327018 | 7.31 | nM | Homo sapiens |