# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4584291 | 4i | EC50 | = | 3.2 | uM | ALA4338387 | 5.50 | nM | Trypanosoma brucei brucei | ||
2. | ALA4584291 | 4i | EC50 | = | 4.8 | uM | ALA4338386 | 5.32 | nM | Trypanosoma brucei brucei | ||
3. | ALA4584291 | 4i | K | = | 3030 | 10'3/M/min | ALA4338385 | 10'3/M/min | Homo sapiens | |||
4. | ALA4584291 | 4i | Ki | = | 0.6 | nM | ALA4338384 | 9.22 | nM | Homo sapiens | ||
5. | ALA4584291 | 4i | INH | = | 85 | % | ALA4338379 | % | Trypanosoma brucei rhodesiense | |||
6. | ALA4584291 | 4i | Ki | = | 0.029 | nM | ALA4338382 | 10.54 | nM | Trypanosoma brucei rhodesiense | ||
7. | ALA4584291 | 4i | Kinact | = | 0.001 | /min | ALA4338381 | /min | Trypanosoma brucei rhodesiense | |||
8. | ALA4584291 | 4i | K | = | 29300 | 10'3/M/min | ALA4338383 | 10'3/M/min | Trypanosoma brucei rhodesiense | |||
9. | ALA4584291 | 4i | Kinact | = | 0.002 | /min | ALA4338378 | /min | Homo sapiens |