| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4585089 | 24 | t1/2 | = | 33.7 | min | ALA5236802 | hr | ||||
| 2. | ALA4585089 | 24 | t1/2 | > | 3 | hr | ALA5236801 | hr | ||||
| 3. | ALA4585089 | 24 | t1/2 | = | 75.7 | min | ALA5236800 | hr | ||||
| 4. | ALA4585089 | 24 | Activity | = | 50 | % | ALA5236794 | % | Homo sapiens | |||
| 5. | ALA4585089 | 24 | t1/2 | = | 1.5 | hr | ALA5236791 | hr | ||||
| 6. | ALA4585089 | 24 | EC50 | = | 10 | nM | ALA5236784 | 8.00 | nM | Homo sapiens | ||
| 7. | ALA4585089 | 24 | IC50 | = | 21 | nM | ALA5236775 | 7.68 | nM | Homo sapiens | ||
| 8. | ALA4585089 | 24 | t1/2 | = | 2.6 | hr | ALA5236696 | hr | ||||
| 9. | ALA4585089 | 24 | INH | 0 | ALA4339143 | Active | % | Mus musculus | ||||
| 10. | ALA4585089 | 24 | Activity | 0 | ALA4339142 | Active | Mus musculus | |||||
| 11. | ALA4585089 | 24 | Activity | 0 | ALA4339141 | Active | Mus musculus | |||||
| 12. | ALA4585089 | 24 | Activity | 0 | ALA4339140 | Active | Mus musculus | |||||
| 13. | ALA4585089 | 24 | Ratio | > | 3 | ALA4339139 | ||||||
| 14. | ALA4585089 | 24 | Ratio | > | 2 | ALA4339138 | ||||||
| 15. | ALA4585089 | 24 | F | = | 28 | % | ALA4339137 | % | ||||
| 16. | ALA4585089 | 24 | t1/2 | = | 1.5 | hr | ALA4339136 | hr | ||||
| 17. | ALA4585089 | 24 | Vd | = | 0.33 | L/Kg | ALA4339135 | L.kg-1 | ||||
| 18. | ALA4585089 | 24 | CL | = | 3.65 | ml/min.kg | ALA4339134 | mL.min-1.kg-1 | ||||
| 19. | ALA4585089 | 24 | AUC | = | 26 | uM.hr | ALA4339133 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 20. | ALA4585089 | 24 | Cmax | = | 5.6 | uM | ALA4339132 | nM |
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