# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4587165 | 32 | Imax | = | 30.2 | % | ALA4481261 | % | Homo sapiens | |||
2. | ALA4587165 | 32 | Drug degradation | < | 15 | % | ALA4481216 | % | ||||
3. | ALA4587165 | 32 | Drug degradation | < | 15 | % | ALA4481217 | % | ||||
4. | ALA4587165 | 32 | t1/2 | = | 54 | min | ALA4481218 | hr | ||||
5. | ALA4587165 | 32 | t1/2 | > | 225 | min | ALA4481219 | hr | ||||
6. | ALA4587165 | 32 | Drug degradation | < | 15 | % | ALA4481220 | % | ||||
7. | ALA4587165 | 32 | Drug degradation | < | 15 | % | ALA4481222 | % | ||||
8. | ALA4587165 | 32 | t1/2 | = | 86 | min | ALA4481221 | hr | ||||
9. | ALA4587165 | 32 | t1/2 | > | 1022 | min | ALA4481223 | hr | ||||
10. | ALA4587165 | 32 | Imax | = | 62.4 | % | ALA4481225 | % | Homo sapiens | |||
11. | ALA4587165 | 32 | Imax | = | 82.8 | % | ALA4481226 | % | Homo sapiens | |||
12. | ALA4587165 | 32 | INH | 0 | ALA4481227 | Active | % | Homo sapiens | ||||
13. | ALA4587165 | 32 | INH | 0 | ALA4481228 | Not Active | % | Homo sapiens | ||||
14. | ALA4587165 | 32 | Imax | = | 86.8 | % | ALA4481231 | % | Homo sapiens | |||
15. | ALA4587165 | 32 | IC50 | = | 25.5 | nM | ALA4481230 | 7.59 | nM | Homo sapiens | ||
16. | ALA4587165 | 32 | IC50 | > | 3 | uM | ALA4481229 | nM | Homo sapiens |