| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4587475 | 8i | Cmin | = | 1.7 | uM | ALA4400406 | uM | ||||
| 2. | ALA4587475 | 8i | Tmin | = | 23.8 | hr | ALA4400407 | hr | ||||
| 3. | ALA4587475 | 8i | Ratio | > | 30 | ALA4400408 | ||||||
| 4. | ALA4587475 | 8i | Activity | 0 | ALA4400385 | Not Active | Mus musculus | |||||
| 5. | ALA4587475 | 8i | Activity | 0 | ALA4400405 | Not Active | Mus musculus | |||||
| 6. | ALA4587475 | 8i | Cp | = | 1661 | nM | ALA4400404 | nM | ||||
| 7. | ALA4587475 | 8i | t1/2 | = | 4.7 | hr | ALA4400403 | hr | ||||
| 8. | ALA4587475 | 8i | AUC | = | 330 | uM.hr | ALA4400402 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA4587475 | 8i | Tmax | = | 7 | hr | ALA4400401 | hr | ||||
| 10. | ALA4587475 | 8i | Cmax | = | 28 | uM | ALA4400400 | nM | ||||
| 11. | ALA4587475 | 8i | Cp | = | 140 | nM | ALA4400399 | nM | ||||
| 12. | ALA4587475 | 8i | t1/2 | = | 8.5 | hr | ALA4400398 | hr | ||||
| 13. | ALA4587475 | 8i | AUC | = | 18 | uM.hr | ALA4400397 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 14. | ALA4587475 | 8i | Tmax | = | 0.25 | hr | ALA4400396 | hr | ||||
| 15. | ALA4587475 | 8i | Cmax | = | 6.6 | uM | ALA4400395 | nM | ||||
| 16. | ALA4587475 | 8i | Activity | = | 88 | % | ALA4400394 | % | Homo sapiens | |||
| 17. | ALA4587475 | 8i | permeability | = | 246 | nm/s | ALA4400393 | nm/s | ||||
| 18. | ALA4587475 | 8i | permeability | = | 1624 | nm/s | ALA4400391 | nm/s | ||||
| 19. | ALA4587475 | 8i | permeability | = | 20 | nm/s | ALA4400392 | nm/s | ||||
| 20. | ALA4587475 | 8i | permeability | = | 845 | nm/s | ALA4400390 | nm/s |
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