Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Comment	Assay	Assay Organism
1.	Gefitinib-based PROTAC 3	PROTAC3	DC50	=	11.7	nM	ALA5160878		nM	Homo sapiens
2.	Gefitinib-based PROTAC 3	PROTAC3	Emax	=	96.6	%	ALA5137697		%	Homo sapiens
3.	Gefitinib-based PROTAC 3	PROTAC3	DC50	=	22.3	nM	ALA5137696		nM	Homo sapiens
4.	Gefitinib-based PROTAC 3	PROTAC3	Emax	=	98.9	%	ALA5137695		%	Homo sapiens
5.	Gefitinib-based PROTAC 3	PROTAC3	DC50	=	11.7	nM	ALA5137694		nM	Homo sapiens
6.	Gefitinib-based PROTAC 3	PROTAC3	DC50	=	12	nM	ALA5136274		nM	Homo sapiens
7.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA5136273	NA		Homo sapiens
8.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380798	Active		Homo sapiens
9.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380758	Not Active		Homo sapiens
10.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380757	Not Active		Homo sapiens
11.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380756	Active		Homo sapiens
12.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380755	Active		Homo sapiens
13.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380748	Active		Homo sapiens
14.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380747	Active		Homo sapiens
15.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380746	Active		Homo sapiens
16.	Gefitinib-based PROTAC 3	PROTAC3	Activity		0		ALA4380745	Active		Homo sapiens
17.	Gefitinib-based PROTAC 3	PROTAC3	DC50	=	11.7	nM	ALA4710101		nM	Homo sapiens
18.	Gefitinib-based PROTAC 3	PROTAC3	Therm_solubility	=	1.23	uM	ALA5105246		nM