# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4588443 | 27o; VU6001376 | INH | = | 76 | % | ALA4310077 | % | Homo sapiens | |||
2. | ALA4588443 | 27o; VU6001376 | Activity | 0 | ALA4310076 | Not Active | Rattus norvegicus | |||||
3. | ALA4588443 | 27o; VU6001376 | Activity | 0 | ALA4310075 | Not Active | Rattus norvegicus | |||||
4. | ALA4588443 | 27o; VU6001376 | Activity | 0 | ALA4310074 | Not Active | Rattus norvegicus | |||||
5. | ALA4588443 | 27o; VU6001376 | Activity | 0 | ALA4310073 | Not Active | Rattus norvegicus | |||||
6. | ALA4588443 | 27o; VU6001376 | Activity | 0 | ALA4310072 | Not Active | Rattus norvegicus | |||||
7. | ALA4588443 | 27o; VU6001376 | Activity | 0 | ALA4310071 | Not Active | Homo sapiens | |||||
8. | ALA4588443 | 27o; VU6001376 | Kp | = | 0.23 | ALA4310070 | ||||||
9. | ALA4588443 | 27o; VU6001376 | Ratio | = | 1.9 | ALA4310069 | ||||||
10. | ALA4588443 | 27o; VU6001376 | permeability | = | 5.4 | ucm/s | ALA4310068 | ucm/s | ||||
11. | ALA4588443 | 27o; VU6001376 | permeability | = | 2.9 | ucm/s | ALA4310067 | ucm/s | ||||
12. | ALA4588443 | 27o; VU6001376 | IC50 | > | 30 | uM | ALA4310066 | nM | Homo sapiens | |||
13. | ALA4588443 | 27o; VU6001376 | IC50 | > | 30 | uM | ALA4310065 | nM | Homo sapiens | |||
14. | ALA4588443 | 27o; VU6001376 | IC50 | > | 30 | uM | ALA4310064 | nM | Homo sapiens | |||
15. | ALA4588443 | 27o; VU6001376 | Drug uptake | = | 46 | nM | ALA4310063 | nM | ||||
16. | ALA4588443 | 27o; VU6001376 | Drug uptake | = | 252 | nM | ALA4310061 | nM | ||||
17. | ALA4588443 | 27o; VU6001376 | Cp | = | 1120 | nM | ALA4310059 | nM | ||||
18. | ALA4588443 | 27o; VU6001376 | Activity | 0 | ALA4310058 | Active | Rattus norvegicus | |||||
19. | ALA4588443 | 27o; VU6001376 | Kp | = | 0.4 | ALA4310053 | ||||||
20. | ALA4588443 | 27o; VU6001376 | Drug uptake | = | 107 | ng/g | ALA4310052 | ng/g |