# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4591047 | 6s | IC50 | = | 0.081 | uM | ALA4373082 | 7.09 | nM | Homo sapiens | ||
2. | ALA4591047 | 6s | IC50 | > | 500 | uM | ALA4373083 | nM | Homo sapiens | |||
3. | ALA4591047 | 6s | IC50 | > | 500 | uM | ALA4373084 | nM | Homo sapiens | |||
4. | ALA4591047 | 6s | IC50 | > | 500 | uM | ALA4373085 | nM | Homo sapiens | |||
5. | ALA4591047 | 6s | IC50 | = | 32.3 | uM | ALA4373086 | 4.49 | nM | Homo sapiens | ||
6. | ALA4591047 | 6s | IC50 | > | 500 | uM | ALA4373087 | nM | Homo sapiens | |||
7. | ALA4591047 | 6s | Ratio IC50 | > | 5000 | ALA4373088 | ||||||
8. | ALA4591047 | 6s | Ratio IC50 | > | 5000 | ALA4373089 | ||||||
9. | ALA4591047 | 6s | Ratio IC50 | > | 5000 | ALA4373090 | Homo sapiens | |||||
10. | ALA4591047 | 6s | Ratio IC50 | > | 5000 | ALA4373091 | ||||||
11. | ALA4591047 | 6s | Activity | 0 | ALA4373092 | Active | Mus musculus | |||||
12. | ALA4591047 | 6s | INH | 0 | ALA4373093 | Active | % | |||||
13. | ALA4591047 | 6s | INH | 0 | ALA4373094 | Not Active | % | |||||
14. | ALA4591047 | 6s | Activity | 0 | ALA4373097 | Dose-dependent effect | Mus musculus | |||||
15. | ALA4591047 | 6s | Activity | 0 | ALA4373100 | Non-Toxic | ||||||
16. | ALA4591047 | 6s | t1/2 | = | 1.4 | hr | ALA4373101 | hr | ||||
17. | ALA4591047 | 6s | Tmax | = | 0.53 | hr | ALA4373102 | hr | ||||
18. | ALA4591047 | 6s | Cmax | = | 511 | ng/ml | ALA4373103 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
19. | ALA4591047 | 6s | AUC | = | 646 | hr.ng/ml | ALA4373104 | ng.hr.mL-1 | ||||
20. | ALA4591047 | 6s | BPR | = | 0.56 | ALA4373105 |