| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4591137 | 4 | t1/2 | = | 1.9 | hr | ALA4308778 | hr | ||||
| 2. | ALA4591137 | 4 | Ct | = | 0.001 | uM | ALA4308777 | uM | ||||
| 3. | ALA4591137 | 4 | Cp | = | 8.7 | uM | ALA4308774 | uM | ||||
| 4. | ALA4591137 | 4 | Activity | = | -87 | % | ALA4308772 | % | Mus musculus | |||
| 5. | ALA4591137 | 4 | AUC | = | 51.5 | uM.hr | ALA4308771 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 6. | ALA4591137 | 4 | Tmax | = | 0.3 | hr | ALA4308770 | hr | ||||
| 7. | ALA4591137 | 4 | Cmax | = | 17.3 | uM | ALA4308769 | nM | ||||
| 8. | ALA4591137 | 4 | Fu | = | 0.9 | % | ALA4308768 | |||||
| 9. | ALA4591137 | 4 | Fu | = | 0.4 | % | ALA4308767 | |||||
| 10. | ALA4591137 | 4 | t1/2 | = | 31 | min | ALA4308766 | hr | ||||
| 11. | ALA4591137 | 4 | t1/2 | = | 10 | min | ALA4308765 | hr | ||||
| 12. | ALA4591137 | 4 | Stability | = | 78 | % | ALA4308763 | % | ||||
| 13. | ALA4591137 | 4 | Stability | = | 53 | % | ALA4308762 | % | ||||
| 14. | ALA4591137 | 4 | Emax | = | 350 | % | ALA4308761 | % | Homo sapiens | |||
| 15. | ALA4591137 | 4 | EC50 | = | 2000 | nM | ALA4308760 | 5.70 | nM | Homo sapiens | ||
| 16. | ALA4591137 | 4 | IC50 | = | 43000 | nM | ALA4308758 | 4.37 | nM | Homo sapiens | ||
| 17. | ALA4591137 | 4 | IC50 | = | 70 | nM | ALA4308759 | 7.16 | nM | Homo sapiens |
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