| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  LY 3200882 | LY-3200882 | F | = | 45.6 | % | ALA4769715 | % | ||||
| 2. | LY 3200882 | LY-3200882 | AUC | = | 943.9 | hr.ng/ml | ALA4769714 | ng.hr.mL-1 | ||||
| 3. | LY 3200882 | LY-3200882 | Cmax | = | 747 | ng/ml | ALA4769713 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 4. | LY 3200882 | LY-3200882 | t1/2 | = | 1.1 | hr | ALA4769712 | hr | ||||
| 5. | LY 3200882 | LY-3200882 | AUC | = | 211.7 | hr.ng/ml | ALA4769711 | ng.hr.mL-1 | ||||
| 6. | LY 3200882 | LY-3200882 | Vdss | = | 2.3 | L/Kg | ALA4769710 | L.kg-1 | ||||
| 7. | LY 3200882 | LY-3200882 | CL | = | 5.2 | L/hr/kg | ALA4769709 | mL.min-1.kg-1 | ||||
| 8. | LY 3200882 | LY-3200882 | t1/2 | = | 0.4 | hr | ALA4769708 | hr | ||||
| 9. | LY 3200882 | LY-3200882 | IC50 | = | 82.9 | nM | ALA4769707 | 7.08 | nM | Mus musculus | ||
| 10. | LY 3200882 | LY-3200882 | IC50 | = | 38.2 | nM | ALA4769705 | 7.42 | nM | Homo sapiens | ||
| 11. | LY 3200882 | LY-3200882 | Activity | 0 | ALA4625385 | Non-Toxic | ||||||
| 12. | LY 3200882 | LY-3200882 | AUC | = | 1658 | ng.hr/ml | ALA4625379 | ng.hr.mL-1 | ||||
| 13. | LY 3200882 | LY-3200882 | AUC | = | 4864 | ng.hr/ml | ALA4625378 | ng.hr.mL-1 | ||||
| 14. | LY 3200882 | LY-3200882 | AUC | = | 20232 | ng.hr/ml | ALA4625376 | ng.hr.mL-1 | ||||
| 15. | LY 3200882 | LY-3200882 | AUC | = | 9949 | ng.hr/ml | ALA4625375 | ng.hr.mL-1 | ||||
| 16. | LY 3200882 | LY-3200882 | T/C | = | 36 | % | ALA4625373 | % | Mus musculus | |||
| 17. | LY 3200882 | LY-3200882 | T/C | = | 57 | % | ALA4625372 | % | Mus musculus | |||
| 18. | LY 3200882 | LY-3200882 | TGI | = | 64 | % | ALA5133861 | % | ||||
| 19. | LY 3200882 | LY-3200882 | TGI | = | 42.5 | % | ALA5133860 | % | ||||
| 20. | LY 3200882 | LY-3200882 | AUC | = | 4864.4 | hr.ng/ml | ALA5133858 | ng.hr.mL-1 |
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