# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4632744 | 2a, diastereomer 1 | Stability | 0 | ALA4623591 | Unstable | % | Homo sapiens | ||||
2. | ALA4632744 | 2a, diastereomer 1 | Stability | 0 | ALA4623591 | Unstable | % | Homo sapiens | ||||
3. | ALA4632744 | 2a, diastereomer 1 | Activity | 0 | ALA4623582 | Not Active | Mus musculus | |||||
4. | ALA4632744 | 2a, diastereomer 1 | Activity | 0 | ALA4623582 | Not Active | Mus musculus | |||||
5. | ALA4632744 | 2a, diastereomer 1 | permeability | 0 | ALA4623590 | Bld | ||||||
6. | ALA4632744 | 2a, diastereomer 1 | permeability | 0 | ALA4623590 | Bld | ||||||
7. | ALA4632744 | 2a, diastereomer 1 | Drug metabolism | 0 | ALA4623589 | Metabolite_Detected | ||||||
8. | ALA4632744 | 2a, diastereomer 1 | Drug metabolism | 0 | ALA4623589 | Metabolite_Detected | ||||||
9. | ALA4632744 | 2a, diastereomer 1 | Ki | = | 24.5 | uM | ALA4623588 | 4.61 | nM | Homo sapiens | ||
10. | ALA4632744 | 2a, diastereomer 1 | Ki | = | 9.68 | uM | ALA4623588 | 5.01 | nM | Homo sapiens | ||
11. | ALA4632744 | 2a, diastereomer 1 | Stability | 0 | ALA4623586 | Stable | % | Homo sapiens | ||||
12. | ALA4632744 | 2a, diastereomer 1 | Stability | 0 | ALA4623586 | Stable | % | Homo sapiens | ||||
13. | ALA4632744 | 2a, diastereomer 1 | t1/2 | > | 5000 | min | ALA4623585 | hr | ||||
14. | ALA4632744 | 2a, diastereomer 1 | t1/2 | > | 5000 | min | ALA4623585 | hr | ||||
15. | ALA4632744 | 2a, diastereomer 1 | Kd | > | 10 | uM | ALA4623583 | nM | Mus musculus | |||
16. | ALA4632744 | 2a, diastereomer 1 | Kd | > | 10 | uM | ALA4623583 | nM | Mus musculus |