# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4633573 | rac-6e | Drug metabolism | 0 | ALA4623830 | Metabolite_Notdetected | ||||||
2. | ALA4633573 | rac-6e | Activity | = | 41.2 | % | ALA4623829 | % | Homo sapiens | |||
3. | ALA4633573 | rac-6e | INH | = | 0 | % | ALA4623828 | % | Homo sapiens | |||
4. | ALA4633573 | rac-6e | INH | > | 90 | % | ALA4623827 | % | Homo sapiens | |||
5. | ALA4633573 | rac-6e | Stability | = | 54 | % | ALA4623826 | % | ||||
6. | ALA4633573 | rac-6e | Therm_solubility | = | 250 | uM | ALA4623825 | nM | ||||
7. | ALA4633573 | rac-6e | Papp | > | 50 | 10'-6 cm/s | ALA4623824 | 10'-6 cm/s | ||||
8. | ALA4633573 | rac-6e | logD | = | 2.1 | ALA4623823 | ||||||
9. | ALA4633573 | rac-6e | IC50 | > | 100000 | nM | ALA4623822 | nM | Homo sapiens | |||
10. | ALA4633573 | rac-6e | IC50 | = | 100 | nM | ALA4623821 | 7.00 | nM | Mus musculus | ||
11. | ALA4633573 | rac-6e | IC50 | = | 28 | nM | ALA4623820 | 7.55 | nM | Homo sapiens | ||
12. | ALA4633573 | rac-6e | IC50 | = | 63000 | nM | ALA4623819 | 4.20 | nM | Homo sapiens | ||
13. | ALA4633573 | rac-6e | IC50 | = | 13000 | nM | ALA4623818 | 4.89 | nM | Homo sapiens |