# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4634770 | 5l; VU6017649 | K(p,uu,brain) | = | 3.88 | ALA4610698 | ||||||
2. | ALA4634770 | 5l; VU6017649 | Kp | = | 1.55 | ALA4610697 | ||||||
3. | ALA4634770 | 5l; VU6017649 | Fu | = | 0.005 | ALA4610696 | ||||||
4. | ALA4634770 | 5l; VU6017649 | Fu | = | 0.007 | ALA4610695 | ||||||
5. | ALA4634770 | 5l; VU6017649 | Fu | = | 0.002 | ALA4610694 | ||||||
6. | ALA4634770 | 5l; VU6017649 | CL | = | 55 | ml/min.kg | ALA4610693 | mL.min-1.kg-1 | ||||
7. | ALA4634770 | 5l; VU6017649 | CL | = | 120 | ml/min.kg | ALA4610692 | mL.min-1.kg-1 | ||||
8. | ALA4634770 | 5l; VU6017649 | EC50 | = | 379 | nM | ALA4610689 | 6.42 | nM | Homo sapiens | ||
9. | ALA4634770 | 5l; VU6017649 | %max | = | 86 | % | ALA4610690 | % | Homo sapiens | |||
10. | ALA4634770 | 5l; VU6017649 | EC50 | = | 226 | nM | ALA4610691 | 6.65 | nM | Rattus norvegicus |