| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4634860 | 1 | Activity | > | 5 | uM | ALA4727499 | uM | ||||
| 2. | ALA4634860 | 1 | Activity | < | 0.001 | uM | ALA4727498 | uM | ||||
| 3. | ALA4634860 | 1 | F | = | 75 | % | ALA4727497 | % | ||||
| 4. | ALA4634860 | 1 | beta t1/2 | = | 4 | hr | ALA4727496 | hr | ||||
| 5. | ALA4634860 | 1 | Vdss | = | 5.1 | L/Kg | ALA4727495 | L.kg-1 | ||||
| 6. | ALA4634860 | 1 | CL | = | 23 | ml/min.kg | ALA4727494 | mL.min-1.kg-1 | ||||
| 7. | ALA4634860 | 1 | Cmax | = | 3230 | nM | ALA4727493 | nM | ||||
| 8. | ALA4634860 | 1 | AUC | = | 29600 | hr.nM | ALA4727492 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA4634860 | 1 | IC50 | = | 1 | uM | ALA4727489 | 6.00 | nM | Homo sapiens | ||
| 10. | ALA4634860 | 1 | IC50 | < | 0.001 | uM | ALA4727488 | nM | Homo sapiens | |||
| 11. | ALA4634860 | 1 | IC50 | < | 0.001 | uM | ALA4727486 | nM | Homo sapiens | |||
| 12. | ALA4634860 | 1 | IC50 | = | 1.2 | uM | ALA4727485 | 5.92 | nM | Mus musculus | ||
| 13. | ALA4634860 | 1 | IC50 | = | 0.004 | uM | ALA4727484 | 8.40 | nM | Mus musculus | ||
| 14. | ALA4634860 | 1 | IC50 | = | 0.068 | uM | ALA4622222 | 7.17 | nM | Homo sapiens |
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