# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4635478 | 9A | fIC50 | = | 3 | nM | ALA4622180 | nM | ||||
2. | ALA4635478 | 9A | fIC50 | = | 3 | nM | ALA4622179 | nM | Homo sapiens | |||
3. | ALA4635478 | 9A | Ratio IC50 | = | 1 | ALA4622216 | Homo sapiens | |||||
4. | ALA4635478 | 9A | Ratio IC50 | = | 1 | ALA4622215 | Homo sapiens | |||||
5. | ALA4635478 | 9A | IC50 | > | 137 | uM | ALA4622213 | nM | Homo sapiens | |||
6. | ALA4635478 | 9A | IC50 | > | 137 | uM | ALA4622211 | nM | Homo sapiens | |||
7. | ALA4635478 | 9A | Kd | = | 0.12 | uM | ALA4622191 | 6.92 | nM | Homo sapiens | ||
8. | ALA4635478 | 9A | Ratio | = | 1.35 | ALA4622190 | ||||||
9. | ALA4635478 | 9A | IC20 | = | 0.9 | uM | ALA4622189 | uM | Homo sapiens | |||
10. | ALA4635478 | 9A | IC50 | = | 2.9 | uM | ALA4622189 | 5.54 | nM | Homo sapiens | ||
11. | ALA4635478 | 9A | Ratio | = | 1 | ALA4622188 | Homo sapiens | |||||
12. | ALA4635478 | 9A | CLH | = | 15 | uL/min | ALA4622187 | uL/min | ||||
13. | ALA4635478 | 9A | CLH | = | 3.3 | uL/min | ALA4622186 | uL/min | ||||
14. | ALA4635478 | 9A | solubility | = | 31 | ug ml-1 | ALA4622185 | ug.mL-1 | ||||
15. | ALA4635478 | 9A | logD | = | 3.9 | ALA4622184 | ||||||
16. | ALA4635478 | 9A | Activity | > | 50 | % | ALA4622183 | % | Mus musculus | |||
17. | ALA4635478 | 9A | Activity | >= | 47 | % | ALA4622182 | % | Mus musculus | |||
18. | ALA4635478 | 9A | Activity | = | 75 | % | ALA4622181 | % | Mus musculus | |||
19. | ALA4635478 | 9A | IC50 | = | 4 | nM | ALA4622180 | 8.40 | nM | |||
20. | ALA4635478 | 9A | PB | = | 96 | pmol | ALA4622219 | pmol |