# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4635767 | 5a, diastereomer 1 | Drug metabolism | 0 | ALA4623592 | Metabolite_Detected | ||||||
2. | ALA4635767 | 5a, diastereomer 1 | Stability | 0 | ALA4623591 | Stable | % | Homo sapiens | ||||
3. | ALA4635767 | 5a, diastereomer 1 | Stability | 0 | ALA4623591 | Stable | % | Homo sapiens | ||||
4. | ALA4635767 | 5a, diastereomer 1 | Activity | 0 | ALA4623582 | Not Active | Mus musculus | |||||
5. | ALA4635767 | 5a, diastereomer 1 | Activity | 0 | ALA4623582 | Not Active | Mus musculus | |||||
6. | ALA4635767 | 5a, diastereomer 1 | permeability | 0 | ALA4623590 | Bld | ||||||
7. | ALA4635767 | 5a, diastereomer 1 | permeability | 0 | ALA4623590 | Bld | ||||||
8. | ALA4635767 | 5a, diastereomer 1 | Drug metabolism | 0 | ALA4623589 | Metabolite_Detected | ||||||
9. | ALA4635767 | 5a, diastereomer 1 | Drug metabolism | 0 | ALA4623589 | Metabolite_Detected | ||||||
10. | ALA4635767 | 5a, diastereomer 1 | Ki | = | 0.74 | uM | ALA4623588 | 6.13 | nM | Homo sapiens | ||
11. | ALA4635767 | 5a, diastereomer 1 | Ki | = | 0.73 | uM | ALA4623588 | 6.14 | nM | Homo sapiens | ||
12. | ALA4635767 | 5a, diastereomer 1 | Stability | 0 | ALA4623586 | Stable | % | Homo sapiens | ||||
13. | ALA4635767 | 5a, diastereomer 1 | Stability | 0 | ALA4623586 | Stable | % | Homo sapiens | ||||
14. | ALA4635767 | 5a, diastereomer 1 | t1/2 | = | 736 | min | ALA4623585 | hr | ||||
15. | ALA4635767 | 5a, diastereomer 1 | t1/2 | = | 2773 | min | ALA4623585 | hr | ||||
16. | ALA4635767 | 5a, diastereomer 1 | Kd | = | 0.49 | uM | ALA4623583 | 6.31 | nM | Mus musculus | ||
17. | ALA4635767 | 5a, diastereomer 1 | Kd | = | 0.23 | uM | ALA4623583 | 6.64 | nM | Mus musculus |