| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4636056 | 9; YA-14-WJ39 | Drug uptake | 0 | ALA4605777 | Active | ||||||
| 2. | ALA4636056 | 9; YA-14-WJ39 | Drug uptake | 0 | ALA4605778 | Active | ||||||
| 3. | ALA4636056 | 9; YA-14-WJ39 | Activity | 0 | ALA4605865 | Non-Toxic | ||||||
| 4. | ALA4636056 | 9; YA-14-WJ39 | INH | 0 | ALA4605864 | Not Active | % | Mus musculus | ||||
| 5. | ALA4636056 | 9; YA-14-WJ39 | INH | 0 | ALA4605863 | Active | % | Mus musculus | ||||
| 6. | ALA4636056 | 9; YA-14-WJ39 | Activity | 0 | ALA4605862 | Active | ||||||
| 7. | ALA4636056 | 9; YA-14-WJ39 | Activity | 0 | ALA4605861 | Active | ||||||
| 8. | ALA4636056 | 9; YA-14-WJ39 | Activity | 0 | ALA4605860 | Active | ||||||
| 9. | ALA4636056 | 9; YA-14-WJ39 | IC50 | = | 2.8 | uM | ALA4605859 | 5.55 | nM | Homo sapiens | ||
| 10. | ALA4636056 | 9; YA-14-WJ39 | IC50 | = | 4.7 | uM | ALA4605858 | 5.33 | nM | Homo sapiens | ||
| 11. | ALA4636056 | 9; YA-14-WJ39 | Ratio | = | 0.13 | ALA4605830 | ||||||
| 12. | ALA4636056 | 9; YA-14-WJ39 | Ratio | = | 0.15 | ALA4605829 | ||||||
| 13. | ALA4636056 | 9; YA-14-WJ39 | F | = | 64 | % | ALA4605779 | % | ||||
| 14. | ALA4636056 | 9; YA-14-WJ39 | Cmax | = | 0.88 | uM | ALA4605781 | nM | ||||
| 15. | ALA4636056 | 9; YA-14-WJ39 | AUC | = | 6.8 | uM.hr | ALA4605780 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 16. | ALA4636056 | 9; YA-14-WJ39 | t1/2 | = | 2.5 | hr | ALA4605782 | hr | ||||
| 17. | ALA4636056 | 9; YA-14-WJ39 | Cmax | = | 1.6 | uM | ALA4605784 | nM | ||||
| 18. | ALA4636056 | 9; YA-14-WJ39 | AUC | = | 2.6 | uM.hr | ALA4605783 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 19. | ALA4636056 | 9; YA-14-WJ39 | t1/2 | = | 1.8 | hr | ALA4605785 | hr | ||||
| 20. | ALA4636056 | 9; YA-14-WJ39 | Vdss | = | 7.8 | L/Kg | ALA4605787 | L.kg-1 |
The page will load shortly, Thanks for your patience!