# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4638732 | 9f | Time | = | 241.7 | s | ALA4604699 | hr | Rattus norvegicus | |||
2. | ALA4638732 | 9f | Time | = | 249.9 | s | ALA4604698 | hr | Rattus norvegicus | |||
3. | ALA4638732 | 9f | IC50 | > | 45 | uM | ALA4604697 | nM | Homo sapiens | |||
4. | ALA4638732 | 9f | IC50 | > | 45 | uM | ALA4604696 | nM | Homo sapiens | |||
5. | ALA4638732 | 9f | BPR | = | 3.79 | ALA4604695 | ||||||
6. | ALA4638732 | 9f | t1/2 | = | 1.07 | hr | ALA4604690 | hr | ||||
7. | ALA4638732 | 9f | AUC | = | 1188 | ng.hr/ml | ALA4604689 | ng.hr.mL-1 | ||||
8. | ALA4638732 | 9f | Cmax | = | 949 | ng/ml | ALA4604688 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
9. | ALA4638732 | 9f | F | = | 50 | % | ALA4604687 | % | ||||
10. | ALA4638732 | 9f | Drug metabolism | = | 40.4 | % | ALA4604686 | % | ||||
11. | ALA4638732 | 9f | Drug metabolism | = | 40.7 | % | ALA4604685 | % | ||||
12. | ALA4638732 | 9f | Ki | = | 0.19 | nM | ALA4604683 | 9.72 | nM | Homo sapiens | ||
13. | ALA4638732 | 9f | Ki | > | 10000 | nM | ALA4604684 | nM | Homo sapiens |