# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4639222 | 4g; VU6016395 | K(p,uu,brain) | = | 0.25 | ALA4610698 | ||||||
2. | ALA4639222 | 4g; VU6016395 | Kp | = | 0.18 | ALA4610697 | ||||||
3. | ALA4639222 | 4g; VU6016395 | Fu | = | 0.011 | ALA4610696 | ||||||
4. | ALA4639222 | 4g; VU6016395 | Fu | = | 0.045 | ALA4610695 | ||||||
5. | ALA4639222 | 4g; VU6016395 | Fu | = | 0.008 | ALA4610694 | ||||||
6. | ALA4639222 | 4g; VU6016395 | CL | = | 9 | ml/min.kg | ALA4610693 | mL.min-1.kg-1 | ||||
7. | ALA4639222 | 4g; VU6016395 | CL | = | 30 | ml/min.kg | ALA4610692 | mL.min-1.kg-1 | ||||
8. | ALA4639222 | 4g; VU6016395 | EC50 | = | 148 | nM | ALA4610689 | 6.83 | nM | Homo sapiens | ||
9. | ALA4639222 | 4g; VU6016395 | %max | = | 80 | % | ALA4610690 | % | Homo sapiens | |||
10. | ALA4639222 | 4g; VU6016395 | EC50 | = | 82 | nM | ALA4610691 | 7.09 | nM | Rattus norvegicus |