| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | CL | = | 26.26 | ml/min.kg | ALA4612973 | mL.min-1.kg-1 | ||||
| 2. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | AUC | = | 1269.5 | hr.ng/ml | ALA4612972 | ng.hr.mL-1 | ||||
| 3. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | t1/2 | = | 2.09 | hr | ALA4612971 | hr | ||||
| 4. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Activity | >= | 50 | % | ALA4612970 | % | ||||
| 5. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Activity | >= | 50 | % | ALA4612969 | % | ||||
| 6. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Activity | 0 | ALA4612968 | Not Active | ||||||
| 7. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Activity | 0 | ALA4612967 | Not Active | ||||||
| 8. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | IC50 | > | 10000 | nM | ALA4612966 | nM | Homo sapiens | |||
| 9. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | IC50 | = | 3350 | nM | ALA4612964 | 5.47 | nM | Homo sapiens | ||
| 10. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | IC50 | = | 7000 | nM | ALA4612965 | 5.16 | nM | Homo sapiens | ||
| 11. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | IC50 | = | 17 | nM | ALA4612962 | 7.77 | nM | Homo sapiens | ||
| 12. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | -1.21 | C | ALA5060944 | C | Homo sapiens | |||
| 13. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | -2.27 | C | ALA5068376 | C | Homo sapiens | |||
| 14. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | -2.22 | C | ALA4650107 | C | Homo sapiens | |||
| 15. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | 0.22 | C | ALA5064660 | C | Homo sapiens | |||
| 16. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | 0.67 | C | ALA5060015 | C | Homo sapiens | |||
| 17. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | 0.18 | C | ALA5067447 | C | Homo sapiens | |||
| 18. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | 0.11 | C | ALA5066518 | C | Homo sapiens | |||
| 19. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | -0.83 | C | ALA5065589 | C | Homo sapiens | |||
| 20. | DCLK1-IN-1 | FMF-03-146-1; DCLK1-IN-1 | Delta TM | = | -0.65 | C | ALA5062802 | C | Homo sapiens |
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