| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4640428 | 26 | Activity | = | 217 | % | ALA4624509 | % | Rattus norvegicus | |||
| 2. | ALA4640428 | 26 | Activity | 0 | ALA4624508 | Non-Toxic | ||||||
| 3. | ALA4640428 | 26 | Activity | 0 | ALA4624507 | Active | Rattus norvegicus | |||||
| 4. | ALA4640428 | 26 | Activity | 0 | ALA4624506 | Active | Rattus norvegicus | |||||
| 5. | ALA4640428 | 26 | Activity | 0 | ALA4624505 | Non-Toxic | ||||||
| 6. | ALA4640428 | 26 | Occ50 | = | 660 | nM | ALA4624504 | nM | Rattus norvegicus | |||
| 7. | ALA4640428 | 26 | INH | < | 20 | % | ALA4624503 | % | Homo sapiens | |||
| 8. | ALA4640428 | 26 | INH | < | 20 | % | ALA4624502 | % | Homo sapiens | |||
| 9. | ALA4640428 | 26 | INH | < | 20 | % | ALA4624501 | % | Homo sapiens | |||
| 10. | ALA4640428 | 26 | INH | < | 20 | % | ALA4624500 | % | Homo sapiens | |||
| 11. | ALA4640428 | 26 | INH | < | 20 | % | ALA4624499 | % | Homo sapiens | |||
| 12. | ALA4640428 | 26 | IC50 | = | 1.5 | uM | ALA4624498 | 5.82 | nM | Homo sapiens | ||
| 13. | ALA4640428 | 26 | BPR | = | 0.59 | ALA4624497 | ||||||
| 14. | ALA4640428 | 26 | Ct | = | 22 | nM | ALA4624496 | nM | ||||
| 15. | ALA4640428 | 26 | Ct | = | 470 | nM | ALA4624495 | nM | ||||
| 16. | ALA4640428 | 26 | permeability | = | 28 | 10'-6 cm/s | ALA4624494 | 10'-6 cm/s | ||||
| 17. | ALA4640428 | 26 | permeability | = | 35 | 10'-6 cm/s | ALA4624493 | 10'-6 cm/s | ||||
| 18. | ALA4640428 | 26 | Kinetic_solubility | > | 100 | uM | ALA4624492 | nM | ||||
| 19. | ALA4640428 | 26 | F | = | 64 | % | ALA4624491 | % | ||||
| 20. | ALA4640428 | 26 | AUC | = | 4416 | ng.hr/ml | ALA4624490 | ng.hr.mL-1 |
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