| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4640857 | 11; OAT-1441 | INH | = | 37 | % | ALA4704020 | % | Homo sapiens | |||
| 2. | ALA4640857 | 11; OAT-1441 | IC50 | = | 22 | uM | ALA4704019 | 4.66 | nM | Homo sapiens | ||
| 3. | ALA4640857 | 11; OAT-1441 | IC50 | = | 59 | nM | ALA4704018 | 7.23 | nM | Mus musculus | ||
| 4. | ALA4640857 | 11; OAT-1441 | IC50 | = | 7 | nM | ALA4704017 | 8.15 | nM | Homo sapiens | ||
| 5. | ALA4640857 | 11; OAT-1441 | IC50 | = | 137 | nM | ALA4704015 | 6.86 | nM | Mus musculus | ||
| 6. | ALA4640857 | 11; OAT-1441 | IC50 | = | 915 | nM | ALA4704014 | 6.04 | nM | Homo sapiens | ||
| 7. | ALA4640857 | 11; OAT-1441 | INH | = | 37 | % | ALA4619035 | % | Rattus norvegicus | |||
| 8. | ALA4640857 | 11; OAT-1441 | IC50 | = | 23000 | nM | ALA4619034 | 4.64 | nM | Homo sapiens | ||
| 9. | ALA4640857 | 11; OAT-1441 | MRT | = | 4.2 | hr | ALA4619033 | hr | ||||
| 10. | ALA4640857 | 11; OAT-1441 | t1/2 | = | 4.2 | hr | ALA4619032 | hr | ||||
| 11. | ALA4640857 | 11; OAT-1441 | Tmax | = | 0.5 | hr | ALA4619031 | hr | ||||
| 12. | ALA4640857 | 11; OAT-1441 | Cmax | = | 3.4 | mg/L | ALA4619030 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 13. | ALA4640857 | 11; OAT-1441 | AUC | = | 22.5 | mg.hr/L | ALA4619029 | ng.hr.mL-1 | ||||
| 14. | ALA4640857 | 11; OAT-1441 | F | = | 41 | % | ALA4619028 | % | ||||
| 15. | ALA4640857 | 11; OAT-1441 | MRT | = | 0.84 | hr | ALA4619027 | hr | ||||
| 16. | ALA4640857 | 11; OAT-1441 | t1/2 | = | 1.1 | hr | ALA4619026 | hr | ||||
| 17. | ALA4640857 | 11; OAT-1441 | Tmax | = | 0.5 | hr | ALA4619025 | hr | ||||
| 18. | ALA4640857 | 11; OAT-1441 | Cmax | = | 3.1 | mg/L | ALA4619024 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 19. | ALA4640857 | 11; OAT-1441 | AUC | = | 3.9 | mg.hr/L | ALA4619023 | ng.hr.mL-1 | ||||
| 20. | ALA4640857 | 11; OAT-1441 | MRT | = | 0.34 | hr | ALA4619022 | hr |
The page will load shortly, Thanks for your patience!