# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4642587 | 1g | MRT | = | 0.239 | hr | ALA4628035 | hr | ||||
2. | ALA4642587 | 1g | AUC | = | 63.7 | ng.hr/ml | ALA4628034 | ng.hr.mL-1 | ||||
3. | ALA4642587 | 1g | AUClast | = | 58.5 | ng.hr/ml | ALA4628033 | ng.hr.mL-1 | ||||
4. | ALA4642587 | 1g | beta t1/2 | = | 0.216 | hr | ALA4628032 | hr | ||||
5. | ALA4642587 | 1g | Vdss | = | 1.72 | L/Kg | ALA4628031 | L.kg-1 | ||||
6. | ALA4642587 | 1g | CL | = | 6.58 | L/hr/kg | ALA4628030 | mL.min-1.kg-1 | ||||
7. | ALA4642587 | 1g | IC50 | = | 13.4 | uM | ALA4628021 | 4.87 | nM | Homo sapiens | ||
8. | ALA4642587 | 1g | IC50 | = | 6 | uM | ALA4628022 | 5.22 | nM | Homo sapiens | ||
9. | ALA4642587 | 1g | IC50 | > | 10 | uM | ALA4628023 | nM | Homo sapiens | |||
10. | ALA4642587 | 1g | IC50 | > | 10 | uM | ALA4628024 | nM | Homo sapiens | |||
11. | ALA4642587 | 1g | IC50 | > | 10 | uM | ALA4628025 | nM | Homo sapiens |