| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4646504 | 36 | INH | = | 35 | % | ALA4614770 | % | Mus musculus | |||
| 2. | ALA4646504 | 36 | INH | = | 43 | % | ALA4614769 | % | Mus musculus | |||
| 3. | ALA4646504 | 36 | F | = | 41 | % | ALA4614766 | % | ||||
| 4. | ALA4646504 | 36 | AUClast | = | 10.8 | uM.hr | ALA4614764 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 5. | ALA4646504 | 36 | MRT | = | 2.1 | hr | ALA4614763 | hr | ||||
| 6. | ALA4646504 | 36 | t1/2 | = | 6.6 | hr | ALA4614762 | hr | ||||
| 7. | ALA4646504 | 36 | Vdss | = | 4.3 | L/Kg | ALA4614761 | L.kg-1 | ||||
| 8. | ALA4646504 | 36 | CL | = | 8 | ml/min.kg | ALA4614760 | mL.min-1.kg-1 | ||||
| 9. | ALA4646504 | 36 | IC50 | = | 0.16 | uM | ALA4614754 | 6.80 | nM | Mus musculus | ||
| 10. | ALA4646504 | 36 | IC50 | = | 0.15 | uM | ALA4614753 | 6.82 | nM | Homo sapiens | ||
| 11. | ALA4646504 | 36 | IC50 | = | 0.024 | uM | ALA4614752 | 7.62 | nM | Homo sapiens |
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