# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4646514 | 18 | t1/2 | = | 0.72 | hr | ALA4622344 | hr | ||||
2. | ALA4646514 | 18 | IC50 | = | 16.8 | uM | ALA4622343 | 4.78 | nM | Homo sapiens | ||
3. | ALA4646514 | 18 | t1/2 | = | 192 | min | ALA4622342 | hr | ||||
4. | ALA4646514 | 18 | t1/2 | = | 108 | min | ALA4622341 | hr | ||||
5. | ALA4646514 | 18 | t1/2 | = | 311 | min | ALA4622340 | hr | ||||
6. | ALA4646514 | 18 | Stability | = | 79.5 | % | ALA4622339 | % | ||||
7. | ALA4646514 | 18 | Stability | = | 89.4 | % | ALA4622338 | % | ||||
8. | ALA4646514 | 18 | Stability | = | 86.8 | % | ALA4622337 | % | ||||
9. | ALA4646514 | 18 | IC50 | > | 3.29 | uM | ALA4622336 | nM | Homo sapiens | |||
10. | ALA4646514 | 18 | IC50 | > | 30 | uM | ALA4622335 | nM | Homo sapiens | |||
11. | ALA4646514 | 18 | IC50 | > | 30 | uM | ALA4622334 | nM | Homo sapiens | |||
12. | ALA4646514 | 18 | IC50 | > | 30 | uM | ALA4622333 | nM | Homo sapiens | |||
13. | ALA4646514 | 18 | IC50 | = | 8.69 | uM | ALA4622332 | 5.06 | nM | Homo sapiens | ||
14. | ALA4646514 | 18 | Stability | = | 106 | % | ALA4622331 | % | ||||
15. | ALA4646514 | 18 | Stability | = | 102 | % | ALA4622330 | % | ||||
16. | ALA4646514 | 18 | IC50 | > | 20 | uM | ALA4622323 | nM | Homo sapiens | |||
17. | ALA4646514 | 18 | Papp | = | 0.09 | ucm/s | ALA4622322 | ucm/s | ||||
18. | ALA4646514 | 18 | t1/2 | = | 4.6 | hr | ALA4622321 | hr | ||||
19. | ALA4646514 | 18 | Cp | = | 163 | nM | ALA4622320 | nM | ||||
20. | ALA4646514 | 18 | Cp | = | 206 | nM | ALA4622319 | nM |