| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4649476 | EU-1180-453 | Activity | 0 | ALA4630152 | Not Active | Rattus norvegicus | |||||
| 2. | ALA4649476 | EU-1180-453 | Activity | 0 | ALA4630151 | Not Active | Rattus norvegicus | |||||
| 3. | ALA4649476 | EU-1180-453 | Drug uptake | = | 2.5 | uM | ALA4630146 | uM | ||||
| 4. | ALA4649476 | EU-1180-453 | Cp | = | 1.83 | uM | ALA4630149 | uM | ||||
| 5. | ALA4649476 | EU-1180-453 | PPB | = | 98.7 | % | ALA4630150 | % | ||||
| 6. | ALA4649476 | EU-1180-453 | BPR | = | 1.4 | ALA4630145 | ||||||
| 7. | ALA4649476 | EU-1180-453 | t1/2 | = | 1.07 | hr | ALA4630144 | hr | ||||
| 8. | ALA4649476 | EU-1180-453 | Cmax | = | 1.83 | uM | ALA4630143 | nM | ||||
| 9. | ALA4649476 | EU-1180-453 | Fu | = | 1.3 | % | ALA4630139 | |||||
| 10. | ALA4649476 | EU-1180-453 | %max | = | 350 | % | ALA4630130 | % | Rattus norvegicus | |||
| 11. | ALA4649476 | EU-1180-453 | %max | = | 350 | % | ALA4630129 | % | Rattus norvegicus | |||
| 12. | ALA4649476 | EU-1180-453 | solubility | = | 74 | uM | ALA4630128 | nM | ||||
| 13. | ALA4649476 | EU-1180-453 | log(activity) | = | -5.7 | ALA4630127 | Rattus norvegicus | |||||
| 14. | ALA4649476 | EU-1180-453 | log(activity) | = | -5.7 | ALA4630126 | Rattus norvegicus | |||||
| 15. | ALA4649476 | EU-1180-453 | pEC50 | = | 5.5 | ALA4630125 | 5.50 | nM | Rattus norvegicus | |||
| 16. | ALA4649476 | EU-1180-453 | pEC50 | = | 5.5 | ALA4630124 | 5.50 | nM | Rattus norvegicus |
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