# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4739883 | 14d | Activity | 0 | ALA4737670 | Non-Toxic | ||||||
2. | ALA4739883 | 14d | TGI | 0 | ALA4737669 | Active | Homo sapiens | |||||
3. | ALA4739883 | 14d | TGI | = | 93.5 | % | ALA4737668 | % | Homo sapiens | |||
4. | ALA4739883 | 14d | MRT | = | 154.15 | min | ALA4737667 | hr | ||||
5. | ALA4739883 | 14d | MRT(t) | = | 113.79 | min | ALA4737666 | min | ||||
6. | ALA4739883 | 14d | AUC | = | 1447.63 | hr.ng/ml | ALA4737665 | ng.hr.mL-1 | ||||
7. | ALA4739883 | 14d | AUCt | = | 1336.16 | hr.ng/ml | ALA4737664 | ng.hr.mL-1 | ||||
8. | ALA4739883 | 14d | Cmax | = | 903 | ng/ml | ALA4737663 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
9. | ALA4739883 | 14d | t1/2 | = | 110.75 | min | ALA4737662 | hr | ||||
10. | ALA4739883 | 14d | INH | 0 | ALA4737661 | Active | % | Homo sapiens | ||||
11. | ALA4739883 | 14d | INH | 0 | ALA4737660 | Active | % | Homo sapiens | ||||
12. | ALA4739883 | 14d | INH | 0 | ALA4737659 | Active | % | |||||
13. | ALA4739883 | 14d | INH | 0 | ALA4737658 | Active | % | |||||
14. | ALA4739883 | 14d | Activity | = | 84 | % | ALA4737657 | % | Homo sapiens | |||
15. | ALA4739883 | 14d | Activity | = | 87 | % | ALA4737656 | % | Homo sapiens | |||
16. | ALA4739883 | 14d | Activity | = | 0.1 | % | ALA4737655 | % | Homo sapiens | |||
17. | ALA4739883 | 14d | Activity | = | 71 | % | ALA4737654 | % | Homo sapiens | |||
18. | ALA4739883 | 14d | Activity | = | 82 | % | ALA4737653 | % | Homo sapiens | |||
19. | ALA4739883 | 14d | Activity | = | 87 | % | ALA4737652 | % | Homo sapiens | |||
20. | ALA4739883 | 14d | Activity | = | 100 | % | ALA4737651 | % | Homo sapiens |