# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4742035 | synthetic Cn2 | Activity | 0 | ALA4720293 | Active | ||||||
2. | ALA4742035 | synthetic Cn2 | Activity | 0 | ALA4720292 | Active | ||||||
3. | ALA4742035 | synthetic Cn2 | Activity | 0 | ALA4720291 | Active | ||||||
4. | ALA4742035 | synthetic Cn2 | Activity | = | 20 | % | ALA4720281 | % | Homo sapiens | |||
5. | ALA4742035 | synthetic Cn2 | delta(V1/2) | = | 10.2 | mV | ALA4720280 | mV | Homo sapiens | |||
6. | ALA4742035 | synthetic Cn2 | Activity | = | 8.2 | ALA4720279 | Homo sapiens | |||||
7. | ALA4742035 | synthetic Cn2 | V1/2 | = | -24.1 | mV | ALA4720278 | mV | Homo sapiens | |||
8. | ALA4742035 | synthetic Cn2 | INH | = | 47.3 | % | ALA4720277 | % | Homo sapiens | |||
9. | ALA4742035 | synthetic Cn2 | INH | 0 | ALA4720276 | Active | % | Homo sapiens | ||||
10. | ALA4742035 | synthetic Cn2 | INH | 0 | ALA4720275 | Active | % | Homo sapiens | ||||
11. | ALA4742035 | synthetic Cn2 | INH | 0 | ALA4720274 | Dose-dependent effect | % | Homo sapiens | ||||
12. | ALA4742035 | synthetic Cn2 | pEC50 | = | 8.2 | ALA4720274 | 8.20 | nM | Homo sapiens | |||
13. | ALA4742035 | synthetic Cn2 | EC50 | = | 6.2 | nM | ALA4720274 | 8.21 | nM | Homo sapiens | ||
14. | ALA4742035 | synthetic Cn2 | EC50 | = | 15.8 | nM | ALA4720273 | 7.80 | nM | Homo sapiens | ||
15. | ALA4742035 | synthetic Cn2 | EC50 | = | 72 | nM | ALA4720273 | 7.14 | nM | Homo sapiens | ||
16. | ALA4742035 | synthetic Cn2 | pEC50 | = | 7.81 | ALA4720273 | 7.81 | nM | Homo sapiens | |||
17. | ALA4742035 | synthetic Cn2 | pEC50 | = | 7.14 | ALA4720273 | 7.14 | nM | Homo sapiens | |||
18. | ALA4742035 | synthetic Cn2 | INH | 0 | ALA4720272 | Not Active | % | Homo sapiens | ||||
19. | ALA4742035 | synthetic Cn2 | INH | 0 | ALA4720271 | Not Active | % | Homo sapiens | ||||
20. | ALA4742035 | synthetic Cn2 | INH | 0 | ALA4720270 | Not Active | % | Homo sapiens |