| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4744083 | 12 | BPR | = | 0.28 | ALA4836422 | ||||||
| 2. | ALA4744083 | 12 | Ct | = | 230 | ng | ALA4836421 | ng | ||||
| 3. | ALA4744083 | 12 | CL | = | 67 | ml/min.kg | ALA4836413 | mL.min-1.kg-1 | ||||
| 4. | ALA4744083 | 12 | t1/2 | = | 0.3 | hr | ALA4836412 | hr | ||||
| 5. | ALA4744083 | 12 | solubility | < | 0.001 | mg/ml | ALA4836411 | ug.mL-1 | ||||
| 6. | ALA4744083 | 12 | solubility | = | 0.163 | mg/ml | ALA4836410 | ug.mL-1 | ||||
| 7. | ALA4744083 | 12 | permeability | = | 50.6 | 10^-6 cm/s | ALA4836409 | 10^-6 cm/s | ||||
| 8. | ALA4744083 | 12 | Cp | = | 808 | ng/ml | ALA4836407 | ng/ml | ||||
| 9. | ALA4744083 | 12 | Drug metabolism | = | 0.852 | umol/ml | ALA4836405 | umol/ml | ||||
| 10. | ALA4744083 | 12 | CLH | = | 0.395 | uL/min | ALA4836404 | uL/min | ||||
| 11. | ALA4744083 | 12 | CLH | = | 1.071 | uL/min | ALA4836403 | uL/min | ||||
| 12. | ALA4744083 | 12 | IC50 | = | 2.4 | nM | ALA4836402 | 8.62 | nM | Homo sapiens | ||
| 13. | ALA4744083 | 12 | IC50 | = | 2.4 | nM | ALA4679436 | 8.62 | nM | Mus musculus | ||
| 14. | ALA4744083 | 12 | IC50 | = | 3.3 | nM | ALA4679434 | 8.48 | nM | Homo sapiens | ||
| 15. | ALA4744083 | 12 | Cp | = | 808 | ng/ml | ALA4679432 | ng/ml | ||||
| 16. | ALA4744083 | 12 | Drug uptake | = | 230 | ng/g | ALA4679431 | ng/g | ||||
| 17. | ALA4744083 | 12 | BPR | = | 0.282 | ALA4679430 | ||||||
| 18. | ALA4744083 | 12 | permeability | = | 50.6 | 10^-6 cm/s | ALA4679429 | 10^-6 cm/s | ||||
| 19. | ALA4744083 | 12 | Activity | 0 | ALA4679428 | Active | ||||||
| 20. | ALA4744083 | 12 | FC | = | 2 | ALA4679427 |
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