# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4745240 | 14a | INH | 0 | ALA4684824 | Active | % | Homo sapiens | ||||
2. | ALA4745240 | 14a | Activity | = | 66.48 | % | ALA4684823 | % | Homo sapiens | |||
3. | ALA4745240 | 14a | GI | = | 57.33 | % | ALA4684822 | % | Homo sapiens | |||
4. | ALA4745240 | 14a | GI | = | 72.88 | % | ALA4684821 | % | Homo sapiens | |||
5. | ALA4745240 | 14a | F | = | 27.8 | % | ALA4684818 | % | ||||
6. | ALA4745240 | 14a | MRT | = | 2.36 | hr | ALA4684817 | hr | ||||
7. | ALA4745240 | 14a | AUC | = | 7200 | ng.hr/ml | ALA4684816 | ng.hr.mL-1 | ||||
8. | ALA4745240 | 14a | Cmax | = | 2170 | ng/ml | ALA4684815 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
9. | ALA4745240 | 14a | Tmax | = | 1 | min | ALA4684814 | hr | ||||
10. | ALA4745240 | 14a | t1/2 | = | 1.63 | min | ALA4684813 | hr | ||||
11. | ALA4745240 | 14a | Activity | 0 | ALA4684812 | Active | Homo sapiens | |||||
12. | ALA4745240 | 14a | INH | 0 | ALA4684811 | Active | % | Homo sapiens | ||||
13. | ALA4745240 | 14a | Activity | 0 | ALA4684810 | Active | Homo sapiens | |||||
14. | ALA4745240 | 14a | Activity | 0 | ALA4684809 | Active | Homo sapiens | |||||
15. | ALA4745240 | 14a | Activity | = | 77.1 | % | ALA4684808 | % | Homo sapiens | |||
16. | ALA4745240 | 14a | Activity | = | 73.08 | % | ALA4684807 | % | Homo sapiens | |||
17. | ALA4745240 | 14a | Activity | 0 | ALA4684806 | Active | Homo sapiens | |||||
18. | ALA4745240 | 14a | Activity | 0 | ALA4684805 | Active | Homo sapiens | |||||
19. | ALA4745240 | 14a | Activity | 0 | ALA4684804 | Active | Homo sapiens | |||||
20. | ALA4745240 | 14a | Activity | 0 | ALA4684803 | Active | Homo sapiens |