| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4747214 | 11; DSM416 | Ratio | = | 0.7 | ALA4706916 | ||||||
| 2. | ALA4747214 | 11; DSM416 | PPB | = | 99.7 | % | ALA4706910 | % | ||||
| 3. | ALA4747214 | 11; DSM416 | PPB | = | 99.2 | % | ALA4706907 | % | ||||
| 4. | ALA4747214 | 11; DSM416 | fAUC | = | 0.09 | uM.hr | ALA4706895 | uM.hr | ||||
| 5. | ALA4747214 | 11; DSM416 | solubility | = | 211 | ug ml-1 | ALA4706893 | ug.mL-1 | ||||
| 6. | ALA4747214 | 11; DSM416 | F | = | 86 | % | ALA4706866 | % | ||||
| 7. | ALA4747214 | 11; DSM416 | fAUC | = | 0.95 | uM.hr | ALA4706861 | uM.hr | ||||
| 8. | ALA4747214 | 11; DSM416 | AUC | = | 318 | uM.hr | ALA4706856 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA4747214 | 11; DSM416 | fCmax | = | 0.11 | uM | ALA4706851 | uM | ||||
| 10. | ALA4747214 | 11; DSM416 | Tmax | = | 2.5 | hr | ALA4706843 | hr | ||||
| 11. | ALA4747214 | 11; DSM416 | fVdss | = | 367 | L/Kg | ALA4706838 | L/Kg | ||||
| 12. | ALA4747214 | 11; DSM416 | Vdss | = | 1.1 | L/Kg | ALA4706833 | L.kg-1 | ||||
| 13. | ALA4747214 | 11; DSM416 | CL free | = | 933 | ml/min.kg | ALA4706828 | mL.min-1.kg-1 | ||||
| 14. | ALA4747214 | 11; DSM416 | CL | = | 2.8 | ml/min.kg | ALA4706823 | mL.min-1.kg-1 | ||||
| 15. | ALA4747214 | 11; DSM416 | AUC | = | 30 | uM.hr | ALA4706818 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 16. | ALA4747214 | 11; DSM416 | t1/2(app) | = | 6.2 | hr | ALA4706813 | hr | ||||
| 17. | ALA4747214 | 11; DSM416 | beta t1/2 | = | 2 | hr | ALA4706811 | hr | ||||
| 18. | ALA4747214 | 11; DSM416 | fAUC | = | 0.41 | uM.hr | ALA4706810 | uM.hr | ||||
| 19. | ALA4747214 | 11; DSM416 | fCmax | = | 0.07 | uM | ALA4706809 | uM | ||||
| 20. | ALA4747214 | 11; DSM416 | AUC | = | 51 | uM.hr | ALA4706808 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 |
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