# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4748423 | 8; Table 1, R4C2 | INH | = | 55 | % | ALA4686877 | % | Homo sapiens | |||
2. | ALA4748423 | 8; Table 1, R4C2 | IC50 | = | 18 | uM | ALA4686875 | 4.75 | nM | Homo sapiens | ||
3. | ALA4748423 | 8; Table 1, R4C2 | IC50 | = | 26 | uM | ALA4686874 | 4.58 | nM | Homo sapiens | ||
4. | ALA4748423 | 8; Table 1, R4C2 | INH | = | 60 | % | ALA4686872 | % | Homo sapiens | |||
5. | ALA4748423 | 8; Table 1, R4C2 | IC50 | = | 460 | uM | ALA4686871 | nM | Homo sapiens | |||
6. | ALA4748423 | 8; Table 1, R4C2 | Activity | 0 | ALA4686869 | Not Active | ||||||
7. | ALA4748423 | 8; Table 1, R4C2 | Activity | 0 | ALA4686867 | Not Active | ||||||
8. | ALA4748423 | 8; Table 1, R4C2 | Activity | 0 | ALA4686866 | Active | ||||||
9. | ALA4748423 | 8; Table 1, R4C2 | Activity | 0 | ALA4686865 | Not Active | ||||||
10. | ALA4748423 | 8; Table 1, R4C2 | Activity | 0 | ALA4686861 | Active | ||||||
11. | ALA4748423 | 8; Table 1, R4C2 | FC | = | 1.13 | ALA4686860 | Homo sapiens | |||||
12. | ALA4748423 | 8; Table 1, R4C2 | Ratio EC50 | = | 5 | ALA4686859 | Homo sapiens | |||||
13. | ALA4748423 | 8; Table 1, R4C2 | Activity | 0 | ALA4686858 | Not Active | Homo sapiens | |||||
14. | ALA4748423 | 8; Table 1, R4C2 | EC50 | = | 10 | uM | ALA4686857 | 5.00 | nM | Homo sapiens | ||
15. | ALA4748423 | 8; Table 1, R4C2 | FC | = | 30 | ALA4686856 | Homo sapiens | |||||
16. | ALA4748423 | 8; Table 1, R4C2 | Emax | = | 260 | % | ALA4686855 | % | Homo sapiens | |||
17. | ALA4748423 | 8; Table 1, R4C2 | Emax | = | 198 | % | ALA4686854 | % | Homo sapiens | |||
18. | ALA4748423 | 8; Table 1, R4C2 | EC50 | = | 11 | uM | ALA4686853 | 4.96 | nM | Homo sapiens | ||
19. | ALA4748423 | 8; Table 1, R4C2 | EC50 | = | 13 | uM | ALA4686852 | 4.89 | nM | |||
20. | ALA4748423 | 8; Table 1, R4C2 | EC50 | = | 3.1 | uM | ALA4686851 | 5.51 | nM |