| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4748638 | 8 | F | = | 36 | % | ALA4727497 | % | ||||
| 2. | ALA4748638 | 8 | beta t1/2 | = | 4.1 | hr | ALA4727496 | hr | ||||
| 3. | ALA4748638 | 8 | Vdss | = | 15 | L/Kg | ALA4727495 | L.kg-1 | ||||
| 4. | ALA4748638 | 8 | CL | = | 98 | ml/min.kg | ALA4727494 | mL.min-1.kg-1 | ||||
| 5. | ALA4748638 | 8 | Cmax | = | 506 | nM | ALA4727493 | nM | ||||
| 6. | ALA4748638 | 8 | AUC | = | 3046 | hr.nM | ALA4727492 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 7. | ALA4748638 | 8 | IC50 | = | 2.7 | uM | ALA4727489 | 5.57 | nM | Homo sapiens | ||
| 8. | ALA4748638 | 8 | IC50 | = | 0.003 | uM | ALA4727488 | 8.52 | nM | Homo sapiens | ||
| 9. | ALA4748638 | 8 | IC50 | = | 0.006 | uM | ALA4727486 | 8.22 | nM | Homo sapiens | ||
| 10. | ALA4748638 | 8 | IC50 | = | 0.84 | uM | ALA4727485 | 6.08 | nM | Mus musculus | ||
| 11. | ALA4748638 | 8 | IC50 | = | 0.038 | uM | ALA4727484 | 7.42 | nM | Mus musculus |
The page will load shortly, Thanks for your patience!