# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4749062 | SM2 | EC50 | = | 0.33 | uM | ALA5124440 | 6.48 | nM | |||
2. | ALA4749062 | SM2 | EC50 | = | 0.96 | uM | ALA5124439 | 6.02 | nM | |||
3. | ALA4749062 | SM2 | EC50 | = | 0.19 | uM | ALA5124438 | 6.72 | nM | Homo sapiens | ||
4. | ALA4749062 | SM2 | EC50 | = | 4.1 | uM | ALA5124437 | 5.39 | nM | Homo sapiens | ||
5. | ALA4749062 | SM2 | EC50 | = | 0.21 | uM | ALA5124436 | 6.68 | nM | Homo sapiens | ||
6. | ALA4749062 | SM2 | EC50 | = | 0.42 | uM | ALA5124435 | 6.38 | nM | Homo sapiens | ||
7. | ALA4749062 | SM2 | EC50 | = | 0.32 | uM | ALA5124434 | 6.50 | nM | Homo sapiens | ||
8. | ALA4749062 | SM2 | Time | = | 8 | day | ALA4700943 | hr | Homo sapiens | |||
9. | ALA4749062 | SM2 | Time | = | 3 | day | ALA4700942 | hr | Homo sapiens | |||
10. | ALA4749062 | SM2 | Activity | 0 | ALA4700941 | Dose-dependent effect | Homo sapiens | |||||
11. | ALA4749062 | SM2 | Cp | = | 7563.3 | fmol/uL | ALA4700940 | fmol/uL | ||||
12. | ALA4749062 | SM2 | Cmax | = | 15126.5 | fmol/uL | ALA4700939 | nM | ||||
13. | ALA4749062 | SM2 | Tmax | = | 16 | hr | ALA4700938 | hr | ||||
14. | ALA4749062 | SM2 | t1/2 | = | 28.8 | hr | ALA4700937 | hr | ||||
15. | ALA4749062 | SM2 | FC | = | 1.5 | ALA4700936 | Homo sapiens | |||||
16. | ALA4749062 | SM2 | Activity | = | 0.63 | % | ALA4700933 | % | Homo sapiens | |||
17. | ALA4749062 | SM2 | Activity | = | 9.97 | % | ALA4700932 | % | Homo sapiens | |||
18. | ALA4749062 | SM2 | Activity | = | 1.81 | % | ALA4700931 | % | Homo sapiens | |||
19. | ALA4749062 | SM2 | Activity | = | 87.6 | % | ALA4700930 | % | Homo sapiens | |||
20. | ALA4749062 | SM2 | Activity | = | 1.41 | % | ALA4700929 | % | Homo sapiens |