# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA281594 | GBR-12909 | Potency | 6.684 | uM | ALA2354254 | active | nM | Homo sapiens | |||
2. | ALA281594 | GBR-12909 | Potency | 22.387 | uM | ALA2114784 | active | nM | Homo sapiens | |||
3. | ALA281594 | GBR-12909 | Potency | 11.22 | uM | ALA2114784 | inconclusive | nM | Homo sapiens | |||
4. | ALA281594 | GBR-12909 | Potency | 5.957 | uM | ALA2354221 | active | nM | Homo sapiens | |||
5. | ALA281594 | GBR-12909 | Potency | 25.119 | uM | ALA3562077 | inconclusive | nM | ||||
6. | ALA281594 | GBR-12909 | Ratio IC50 | = | 0 | ALA3385969 | ||||||
7. | ALA281594 | GBR-12909 | Ratio IC50 | = | 0.4 | ALA3385968 | ||||||
8. | ALA281594 | GBR-12909 | IC50 | = | 190 | nM | ALA3385967 | 6.72 | nM | Homo sapiens | ||
9. | ALA281594 | GBR-12909 | IC50 | = | 1460 | nM | ALA3385966 | 5.84 | nM | Homo sapiens | ||
10. | ALA281594 | GBR-12909 | IC50 | = | 3840 | nM | ALA3385965 | 5.42 | nM | Homo sapiens | ||
11. | ALA281594 | GBR-12909 | INH | = | 29 | % | ALA3385964 | % | Homo sapiens | |||
12. | ALA281594 | GBR-12909 | INH | = | -6 | % | ALA3385963 | % | Homo sapiens | |||
13. | ALA281594 | GBR-12909 | INH | = | 2 | % | ALA3385962 | % | Homo sapiens | |||
14. | ALA281594 | GBR-12909 | Ratio Ki | = | 0.78 | ALA3371726 | ||||||
15. | ALA281594 | GBR-12909 | Ratio Ki | = | 0.04 | ALA3371725 | ||||||
16. | ALA281594 | GBR-12909 | Ki | = | 24.1 | nM | ALA3371724 | 7.62 | nM | Mus musculus | ||
17. | ALA281594 | GBR-12909 | Ki | = | 12 | nM | ALA3371727 | 7.92 | nM | Mus musculus | ||
18. | ALA281594 | GBR-12909 | INH | > | 50 | % | ALA4426163 | % | Homo sapiens | |||
19. | ALA281594 | GBR-12909 | Ki | = | 8.8 | nM | ALA4426160 | 8.06 | nM | Homo sapiens | ||
20. | ALA281594 | GBR-12909 | pIC50 | < | 4.7 | ALA4651403 | No. Measurements = 1 | nM | Severe acute respiratory syndrome coronavirus 2 |