# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4749790 | ent-2a | F | = | 1.3 | % | ALA4676193 | % | ||||
2. | ALA4749790 | ent-2a | t1/2 | = | 0.82 | hr | ALA4676192 | hr | ||||
3. | ALA4749790 | ent-2a | CL | = | 4.7 | L/hr/kg | ALA4676191 | mL.min-1.kg-1 | ||||
4. | ALA4749790 | ent-2a | CL | = | 1.9 | L/hr/kg | ALA4676191 | mL.min-1.kg-1 | ||||
5. | ALA4749790 | ent-2a | CLH | = | 2.8 | L/hr/kg | ALA4676186 | mL.min-1.kg-1 | ||||
6. | ALA4749790 | ent-2a | CLH | = | 1.2 | L/hr/kg | ALA4676186 | mL.min-1.kg-1 | ||||
7. | ALA4749790 | ent-2a | IC50 | 0 | ALA4676184 | Not Determined | Rattus norvegicus | |||||
8. | ALA4749790 | ent-2a | IC50 | = | 34 | nM | ALA4676184 | 7.47 | nM | Rattus norvegicus | ||
9. | ALA4749790 | ent-2a | IC50 | >= | 20 | 10^3nM | ALA4676183 | 10^3nM | Rattus norvegicus | |||
10. | ALA4749790 | ent-2a | IC50 | = | 29 | nM | ALA4676183 | 7.54 | nM | Rattus norvegicus | ||
11. | ALA4749790 | ent-2a | IC50 | >= | 20 | 10^3nM | ALA4676182 | 10^3nM | Homo sapiens | |||
12. | ALA4749790 | ent-2a | IC50 | = | 99 | nM | ALA4676182 | 7.00 | nM | Homo sapiens | ||
13. | ALA4749790 | ent-2a | IC50 | = | 28 | nM | ALA4676182 | 7.55 | nM | Homo sapiens | ||
14. | ALA4749790 | ent-2a | IC50 | >= | 20 | 10^3nM | ALA4676181 | 10^3nM | Homo sapiens | |||
15. | ALA4749790 | ent-2a | IC50 | = | 41 | nM | ALA4676181 | 7.39 | nM | Homo sapiens | ||
16. | ALA4749790 | ent-2a | IC50 | = | 15 | nM | ALA4676181 | 7.82 | nM | Homo sapiens |