| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4751832 | 29 | PPB | = | 99 | % | ALA4715008 | % | ||||
| 2. | ALA4751832 | 29 | Activity | 0 | ALA4715007 | Non-Toxic | ||||||
| 3. | ALA4751832 | 29 | INH | 0 | ALA4715006 | Active | % | |||||
| 4. | ALA4751832 | 29 | IC50 | = | 7.8 | uM | ALA4715005 | 5.11 | nM | Homo sapiens | ||
| 5. | ALA4751832 | 29 | IC50 | > | 10 | uM | ALA4715004 | nM | Homo sapiens | |||
| 6. | ALA4751832 | 29 | IC50 | > | 10 | uM | ALA4715003 | nM | Homo sapiens | |||
| 7. | ALA4751832 | 29 | IC50 | > | 10 | uM | ALA4715002 | nM | Homo sapiens | |||
| 8. | ALA4751832 | 29 | IC50 | > | 10 | uM | ALA4715001 | nM | Homo sapiens | |||
| 9. | ALA4751832 | 29 | IC50 | > | 10 | uM | ALA4715000 | nM | Homo sapiens | |||
| 10. | ALA4751832 | 29 | F | = | 48 | % | ALA4714999 | % | ||||
| 11. | ALA4751832 | 29 | t1/2 | = | 4.6 | hr | ALA4714998 | hr | ||||
| 12. | ALA4751832 | 29 | AUC | = | 2.3 | uM/hr | ALA4714997 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 13. | ALA4751832 | 29 | Vdss | = | 2.7 | L/Kg | ALA4714996 | L.kg-1 | ||||
| 14. | ALA4751832 | 29 | CL | = | 0.49 | L/hr/kg | ALA4714995 | mL.min-1.kg-1 | ||||
| 15. | ALA4751832 | 29 | MRT | = | 5.5 | hr | ALA4714994 | hr | ||||
| 16. | ALA4751832 | 29 | IC50 | = | 22.8 | uM | ALA4714993 | 4.64 | nM | Homo sapiens | ||
| 17. | ALA4751832 | 29 | permeability | = | 14 | 10^-7 cm/s | ALA4714992 | 10^-7 cm/s | ||||
| 18. | ALA4751832 | 29 | solubility | 0 | ALA4714991 | Soluble | ||||||
| 19. | ALA4751832 | 29 | Stabilty | = | 84 | % | ALA4714990 | % | ||||
| 20. | ALA4751832 | 29 | Stabilty | = | 74 | % | ALA4714989 | % |
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