# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4753773 | 107; PROTAC 2 | pIC50 | = | 8.1 | ALA5137714 | 8.10 | nM | ||||
2. | ALA4753773 | 107; PROTAC 2 | pKd | = | 9 | ALA5137713 | 9.00 | nM | Homo sapiens | |||
3. | ALA4753773 | 107; PROTAC 2 | Drug uptake | = | 37.2 | pmol | ALA4735370 | pmol | ||||
4. | ALA4753773 | 107; PROTAC 2 | Drug uptake | = | 4.69 | pmol | ALA4735369 | pmol | ||||
5. | ALA4753773 | 107; PROTAC 2 | GI50 | = | 45 | nM | ALA4735368 | nM | Homo sapiens | |||
6. | ALA4753773 | 107; PROTAC 2 | Kd | < | 1 | nM | ALA4735367 | nM | Homo sapiens |