# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4754247 | 21m; S16 | IC50 | = | 138 | nM | ALA4676505 | 6.86 | nM | Homo sapiens | ||
2. | ALA4754247 | 21m; S16 | IC50 | = | 27 | nM | ALA4676504 | 7.57 | nM | Homo sapiens | ||
3. | ALA4754247 | 21m; S16 | IC50 | > | 5000 | nM | ALA4676502 | nM | ||||
4. | ALA4754247 | 21m; S16 | Activity | = | 575 | % | ALA4676501 | % | Homo sapiens | |||
5. | ALA4754247 | 21m; S16 | Activity | = | 212 | % | ALA4676500 | % | Homo sapiens | |||
6. | ALA4754247 | 21m; S16 | INH | = | 19 | % | ALA4676498 | % | Homo sapiens | |||
7. | ALA4754247 | 21m; S16 | INH | = | 55 | % | ALA4676497 | % | Homo sapiens | |||
8. | ALA4754247 | 21m; S16 | IC50 | > | 5000 | nM | ALA4676496 | nM | Rattus norvegicus | |||
9. | ALA4754247 | 21m; S16 | IC50 | > | 5000 | nM | ALA4676495 | nM | Homo sapiens | |||
10. | ALA4754247 | 21m; S16 | IC50 | > | 5000 | nM | ALA4676494 | nM | Homo sapiens | |||
11. | ALA4754247 | 21m; S16 | IC50 | > | 5000 | nM | ALA4676493 | nM | Homo sapiens | |||
12. | ALA4754247 | 21m; S16 | IC50 | = | 6762 | nM | ALA4676491 | 5.17 | nM | Homo sapiens | ||
13. | ALA4754247 | 21m; S16 | INH | = | 77 | % | ALA4676490 | % | Homo sapiens | |||
14. | ALA4754247 | 21m; S16 | INH | = | 92 | % | ALA4676489 | % | Homo sapiens | |||
15. | ALA4754247 | 21m; S16 | Activity | = | 36 | % | ALA4676488 | % | Homo sapiens | |||
16. | ALA4754247 | 21m; S16 | Activity | = | 25 | % | ALA4676487 | % | Homo sapiens | |||
17. | ALA4754247 | 21m; S16 | IC50 | > | 5000 | nM | ALA4676486 | nM | Homo sapiens | |||
18. | ALA4754247 | 21m; S16 | INH | = | 48 | % | ALA4676483 | % | Homo sapiens | |||
19. | ALA4754247 | 21m; S16 | 2aPTT | = | 107 | uM | ALA4676479 | uM | Homo sapiens | |||
20. | ALA4754247 | 21m; S16 | INH | 0 | ALA4676475 | Dose-dependent effect | % | Homo sapiens |