| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4754486 | 40 | Ki | = | 4.2 | nM | ALA4705223 | 8.38 | nM | Homo sapiens | ||
| 2. | ALA4754486 | 40 | t1/2 | > | 360 | min | ALA4705222 | hr | ||||
| 3. | ALA4754486 | 40 | t1/2 | = | 186.1 | min | ALA4705221 | hr | ||||
| 4. | ALA4754486 | 40 | Stabilty | = | 79.5 | % | ALA4705220 | % | ||||
| 5. | ALA4754486 | 40 | Stabilty | = | 93.7 | % | ALA4705219 | % | ||||
| 6. | ALA4754486 | 40 | Stabilty | = | 99.1 | % | ALA4705218 | % | Sus scrofa | |||
| 7. | ALA4754486 | 40 | Stabilty | = | 42.7 | % | ALA4705217 | % | Bos taurus | |||
| 8. | ALA4754486 | 40 | PPB | = | 99.23 | % | ALA4705216 | % | ||||
| 9. | ALA4754486 | 40 | t1/2 | = | 0.78 | hr | ALA4705215 | hr | ||||
| 10. | ALA4754486 | 40 | Vdss | = | 0.29 | L/Kg | ALA4705214 | L.kg-1 | ||||
| 11. | ALA4754486 | 40 | CL | = | 24.25 | ml/min.kg | ALA4705213 | mL.min-1.kg-1 | ||||
| 12. | ALA4754486 | 40 | AUC | = | 490.65 | nM.hr | ALA4705212 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 13. | ALA4754486 | 40 | AUC | = | 491.78 | nM.hr | ALA4705211 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 14. | ALA4754486 | 40 | Ki | = | 23.3 | nM | ALA4705210 | 7.63 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!