# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4755779 | 31 | BPR | = | 0.4 | ALA4672664 | ||||||
2. | ALA4755779 | 31 | Drug uptake | = | 346 | ng/ml | ALA4672662 | ng/ml | ||||
3. | ALA4755779 | 31 | Cp | = | 831 | ng/ml | ALA4672660 | ng/ml | ||||
4. | ALA4755779 | 31 | t1/2 | < | 4 | min | ALA4672659 | hr | ||||
5. | ALA4755779 | 31 | t1/2 | < | 4 | min | ALA4672658 | hr | ||||
6. | ALA4755779 | 31 | CLH | > | 347 | microL/min/mg | ALA4672657 | mL.min-1.g-1 | ||||
7. | ALA4755779 | 31 | CLH | > | 347 | microL/min/mg | ALA4672656 | mL.min-1.g-1 | ||||
8. | ALA4755779 | 31 | INH | = | 41 | % | ALA4672649 | % | Homo sapiens | |||
9. | ALA4755779 | 31 | INH | = | 43 | % | ALA4672648 | % | Homo sapiens | |||
10. | ALA4755779 | 31 | INH | = | 7 | % | ALA4672647 | % | Homo sapiens | |||
11. | ALA4755779 | 31 | INH | = | 31 | % | ALA4672646 | % | Homo sapiens | |||
12. | ALA4755779 | 31 | INH | = | 28 | % | ALA4672644 | % | Homo sapiens | |||
13. | ALA4755779 | 31 | solubility | = | 92 | uM | ALA4672643 | nM | ||||
14. | ALA4755779 | 31 | IC50 | > | 10000 | nM | ALA4672639 | nM | Homo sapiens | |||
15. | ALA4755779 | 31 | IC50 | > | 10000 | nM | ALA4672637 | nM | Homo sapiens | |||
16. | ALA4755779 | 31 | IC50 | > | 10000 | nM | ALA4672636 | nM | ||||
17. | ALA4755779 | 31 | IC50 | = | 912 | nM | ALA4672634 | 6.04 | nM | Rattus norvegicus | ||
18. | ALA4755779 | 31 | IC50 | = | 56 | nM | ALA4672633 | 7.25 | nM | Homo sapiens | ||
19. | ALA4755779 | 31 | IC50 | = | 3.4 | nM | ALA4672632 | 8.47 | nM | Homo sapiens | ||
20. | ALA4755779 | 31 | IC50 | > | 10000 | nM | ALA4672630 | nM | Homo sapiens |