| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4756563 | 34 | Vdss | = | 1 | L/Kg | ALA4724183 | L.kg-1 | ||||
| 2. | ALA4756563 | 34 | CL | = | 2.9 | ml/min.kg | ALA4724182 | mL.min-1.kg-1 | ||||
| 3. | ALA4756563 | 34 | t1/2 | = | 3.8 | hr | ALA4724181 | hr | ||||
| 4. | ALA4756563 | 34 | AUClast | = | 11 | uM.hr | ALA4724180 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 5. | ALA4756563 | 34 | Cmax | = | 1.7 | uM | ALA4724179 | nM | ||||
| 6. | ALA4756563 | 34 | Tmax | = | 0.08 | hr | ALA4724178 | hr | ||||
| 7. | ALA4756563 | 34 | Vdss | = | 0.4 | L/Kg | ALA4724158 | L.kg-1 | ||||
| 8. | ALA4756563 | 34 | CL | = | 0.8 | ml/min.kg | ALA4724157 | mL.min-1.kg-1 | ||||
| 9. | ALA4756563 | 34 | t1/2 | = | 6.4 | hr | ALA4724156 | hr | ||||
| 10. | ALA4756563 | 34 | Drug uptake(free) | = | 166.1 | nM | ALA4724154 | nM | ||||
| 11. | ALA4756563 | 34 | Drug uptake(free) | = | 157.6 | nM | ALA4724153 | nM | ||||
| 12. | ALA4756563 | 34 | PPB | = | 98.86 | % | ALA4724152 | % | ||||
| 13. | ALA4756563 | 34 | PPB | = | 96.92 | % | ALA4724151 | % | ||||
| 14. | ALA4756563 | 34 | PPB | = | 96.98 | % | ALA4724150 | % | ||||
| 15. | ALA4756563 | 34 | ED50 | = | 5.45 | mg kg-1 | ALA4724149 | mg.kg-1 | Homo sapiens | |||
| 16. | ALA4756563 | 34 | ED50 | = | 6.47 | mg kg-1 | ALA4724148 | mg.kg-1 | Homo sapiens | |||
| 17. | ALA4756563 | 34 | Cp | = | 0.38 | uM | ALA4724147 | uM | ||||
| 18. | ALA4756563 | 34 | Drug uptake | = | 0.2 | uM | ALA4724146 | uM | ||||
| 19. | ALA4756563 | 34 | Activity | = | 23.63 | g | ALA4724145 | g | ||||
| 20. | ALA4756563 | 34 | Activity | = | 0.87 | g | ALA4724144 | g | Homo sapiens |
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