# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4758183 | 13g; VU602229 | Activity | 0 | ALA4737565 | Dose-dependent effect | Rattus norvegicus | |||||
2. | ALA4758183 | 13g; VU602229 | Time | = | 22.2 | s | ALA4737564 | hr | Rattus norvegicus | |||
3. | ALA4758183 | 13g; VU602229 | Time | = | 28.6 | s | ALA4737563 | hr | Rattus norvegicus | |||
4. | ALA4758183 | 13g; VU602229 | Time | = | 36.6 | s | ALA4737562 | hr | Rattus norvegicus | |||
5. | ALA4758183 | 13g; VU602229 | INH | = | 55.4 | % | ALA4737561 | % | Rattus norvegicus | |||
6. | ALA4758183 | 13g; VU602229 | INH | = | 42.6 | % | ALA4737560 | % | Rattus norvegicus | |||
7. | ALA4758183 | 13g; VU602229 | INH | = | 26.5 | % | ALA4737559 | % | Rattus norvegicus | |||
8. | ALA4758183 | 13g; VU602229 | Kinetic_solubility | = | 6.2 | uM | ALA4737558 | nM | ||||
9. | ALA4758183 | 13g; VU602229 | IC50 | > | 10 | uM | ALA4737557 | nM | Homo sapiens | |||
10. | ALA4758183 | 13g; VU602229 | IC50 | > | 10 | uM | ALA4737556 | nM | Homo sapiens | |||
11. | ALA4758183 | 13g; VU602229 | IC50 | > | 10 | uM | ALA4737555 | nM | Homo sapiens | |||
12. | ALA4758183 | 13g; VU602229 | IC50 | > | 10 | uM | ALA4737554 | nM | Homo sapiens | |||
13. | ALA4758183 | 13g; VU602229 | IC50 | > | 10 | uM | ALA4737553 | nM | Rattus norvegicus | |||
14. | ALA4758183 | 13g; VU602229 | K(p,uu,brain) | = | 0.7 | ALA4737552 | ||||||
15. | ALA4758183 | 13g; VU602229 | Kp | = | 0.45 | ALA4737551 | ||||||
16. | ALA4758183 | 13g; VU602229 | Fu | = | 0.028 | ALA4737550 | ||||||
17. | ALA4758183 | 13g; VU602229 | Fu | = | 0.011 | ALA4737549 | ||||||
18. | ALA4758183 | 13g; VU602229 | Fu | = | 0.018 | ALA4737548 | ||||||
19. | ALA4758183 | 13g; VU602229 | %max | = | 108 | % | ALA4737547 | % | Rattus norvegicus | |||
20. | ALA4758183 | 13g; VU602229 | EC50 | = | 33 | nM | ALA4737546 | 7.48 | nM | Rattus norvegicus |