# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4759030 | 12 | CC50 | > | 25 | uM | ALA4731381 | nM | Mus musculus | |||
2. | ALA4759030 | 12 | CC50 | > | 25 | uM | ALA4731379 | nM | Mus musculus | |||
3. | ALA4759030 | 12 | CC50 | > | 25 | uM | ALA4731378 | nM | Homo sapiens | |||
4. | ALA4759030 | 12 | Ratio CC50/EC50 | > | 9.7 | ALA4731375 | ||||||
5. | ALA4759030 | 12 | Ratio CC50/EC50 | > | 5 | ALA4731372 | ||||||
6. | ALA4759030 | 12 | INH | = | 59 | % | ALA4731369 | % | Venezuelan equine encephalitis virus | |||
7. | ALA4759030 | 12 | INH | = | 100 | % | ALA4731368 | % | Venezuelan equine encephalitis virus | |||
8. | ALA4759030 | 12 | INH | 0 | ALA4731367 | Dose-dependent effect | % | Venezuelan equine encephalitis virus | ||||
9. | ALA4759030 | 12 | EC50 | = | 2.7 | uM | ALA4731366 | 5.57 | nM | Venezuelan equine encephalitis virus | ||
10. | ALA4759030 | 12 | EC50 | = | 3.4 | uM | ALA4731363 | 5.47 | nM | Venezuelan equine encephalitis virus | ||
11. | ALA4759030 | 12 | Ratio CC50/EC50 | > | 7.3 | ALA4731362 | ||||||
12. | ALA4759030 | 12 | EC50 | = | 4.5 | uM | ALA4731361 | 5.35 | nM | Venezuelan equine encephalitis virus |