| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4759521 | 17f | INH | = | 67 | % | ALA4667336 | % | Homo sapiens | |||
| 2. | ALA4759521 | 17f | Fu | = | 0.041 | ALA4667334 | ||||||
| 3. | ALA4759521 | 17f | Fu | = | 0.003 | ALA4667333 | ||||||
| 4. | ALA4759521 | 17f | Fu | = | 0.052 | ALA4667332 | ||||||
| 5. | ALA4759521 | 17f | Cmax | = | 8.8 | uM | ALA4667331 | nM | ||||
| 6. | ALA4759521 | 17f | beta t1/2 | = | 6.3 | hr | ALA4667330 | hr | ||||
| 7. | ALA4759521 | 17f | AUC | = | 60.6 | uM.hr | ALA4667329 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 8. | ALA4759521 | 17f | Activity | = | 101 | % | ALA4667328 | % | Homo sapiens | |||
| 9. | ALA4759521 | 17f | Activity | = | 84 | % | ALA4667325 | % | Homo sapiens | |||
| 10. | ALA4759521 | 17f | EC50 | = | 6.1 | uM | ALA4667324 | 5.21 | nM | Homo sapiens | ||
| 11. | ALA4759521 | 17f | EC50 | = | 5.5 | uM | ALA4667323 | 5.26 | nM | Homo sapiens | ||
| 12. | ALA4759521 | 17f | Activity | = | -16 | % | ALA4667322 | % | Homo sapiens | |||
| 13. | ALA4759521 | 17f | Activity | = | -9 | % | ALA4667321 | % | Homo sapiens | |||
| 14. | ALA4759521 | 17f | INH | = | 94 | % | ALA4667320 | % | Homo sapiens | |||
| 15. | ALA4759521 | 17f | Activity | = | -21 | % | ALA4667319 | % | Homo sapiens | |||
| 16. | ALA4759521 | 17f | INH | = | 76 | % | ALA4667318 | % | Homo sapiens | |||
| 17. | ALA4759521 | 17f | INH | = | -32 | % | ALA4667317 | % | Homo sapiens | |||
| 18. | ALA4759521 | 17f | INH | = | 57 | % | ALA4667316 | % | Homo sapiens | |||
| 19. | ALA4759521 | 17f | INH | = | 39 | % | ALA4667315 | % | Homo sapiens | |||
| 20. | ALA4759521 | 17f | INH | = | 7 | % | ALA4667314 | % | Homo sapiens |
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